Target Details
| UniProt AC | P03366 |
|---|---|
| Gene Symbol | gag-pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 group M subtype B (isolate BH10) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC) |
Summary
- Multi-target molecules 580
- Clinical molecules 0
- Avg pChEMBL 7.7
Top Co-occurrence Targets
- env 319 shared
- pol 259 shared
- reverse transcriptase 6 shared
- pol 1 shared
- DHODH 1 shared
Active Molecules (580)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FIGRBQAMMXFIMA
|
6.7 | IC50 | 2 | — | |
KTGXCGWBRPNPJN
|
6.7 | IC50 | 2 | — | |
SNEUVPRZHPSNON
|
6.7 | IC50 | 2 | — | |
ZCMRTFYSMQNOKC
|
6.7 | IC50 | 2 | — | |
JFFZDHWSXQDFFY
|
6.7 | IC50 | 2 | — | |
KWWWAPRSFOPABI
|
6.7 | IC50 | 2 | — | |
LYAZZAPFCMSYCJ
|
6.7 | IC50 | 2 | — | |
ZBRYMJQGTZVHEN
|
6.7 | IC50 | 2 | — | |
NWYOKVNRAZZLMG
|
6.7 | IC50 | 2 | — | |
IKARPARVOYZNHF
|
6.7 | IC50 | 2 | — | |
NRPOYRRCQSGMTG
|
6.7 | IC50 | 2 | — | |
NVNZPDYBQNEBRX
|
6.7 | IC50 | 2 | — | |
PGICMOMWBVXUKZ
|
6.7 | IC50 | 2 | — | |
QHRNKMUAIFHYDI
|
6.7 | IC50 | 2 | — | |
VBJZVMYVUMEGLS
|
6.7 | IC50 | 2 | — | |
VSOOMDQCUKVIFC
|
6.7 | IC50 | 2 | — | |
MWENNCGXKSSEBF
|
6.7 | IC50 | 2 | — | |
LVLYKMQPZNKKHZ
|
6.7 | IC50 | 2 | — | |
LWTPUALMLDLRFE
|
6.7 | IC50 | 2 | — | |
VMLPTJUPIGUEIY
|
6.7 | IC50 | 2 | — | |
DPXBRUSUWOSCSF
|
6.6 | IC50 | 2 | — | |
FKLCIYOEQBQJSS
|
6.6 | IC50 | 2 | — | |
GCJKAPWJHBJEPX
|
6.6 | IC50 | 2 | — | |
OXERMLHLBWPCON
|
6.6 | IC50 | 2 | — | |
POSQQJCPFZCRSB
|
6.6 | IC50 | 2 | — | |
SNZNEMLKKGAZGA
|
6.6 | IC50 | 2 | — | |
YVSYYWQMGXODIQ
|
6.6 | IC50 | 2 | — | |
IQNYCOUCSXHAEB
|
6.6 | IC50 | 2 | — | |
BEDHGLWDRNTRSG
|
6.6 | IC50 | 2 | — | |
HIKOPTDSAVXYGS
|
6.6 | IC50 | 2 | — | |
NUPNETPGMWUZFL
|
6.6 | IC50 | 2 | — | |
RAEHLIVJXCOVLZ
|
6.6 | IC50 | 2 | — | |
XZKUDZNOAWQGAL
|
6.6 | IC50 | 2 | — | |
YFEJBNCFMFTPFP
|
6.6 | IC50 | 2 | — | |
ZZUMQCQQGMHBPQ
|
6.6 | IC50 | 2 | — | |
MUKSMBAVCDPKRC
|
6.6 | IC50 | 2 | — | |
ULBJEZHPUJEVCL
|
6.6 | IC50 | 2 | — | |
ZQSLENRLXSUOFJ
|
6.6 | IC50 | 2 | — | |
NIIDNAOMTQCSGR
|
6.6 | IC50 | 2 | — | |
QNNJBKMUOFJXHX
|
6.6 | IC50 | 2 | — | |
VECCARSSBYBIFI
|
6.6 | IC50 | 2 | — | |
KSEACRWZEWHBII
|
6.6 | IC50 | 2 | — | |
DVBVMVZJNSPCMP
|
6.5 | IC50 | 2 | — | |
PDWANTHUWHWFIR
|
6.5 | IC50 | 2 | — | |
SASUXSFGYXUPHS
|
6.5 | IC50 | 2 | — | |
SDHDKVPVUDEWQJ
|
6.5 | IC50 | 2 | — | |
VWPZVQSMQVKQCI
|
6.5 | IC50 | 2 | — | |
AFCUXPVAIWIPIK
|
6.5 | IC50 | 2 | — | |
NGBSYADTRKVTPO
|
6.5 | IC50 | 2 | — | |
NXORHDRQGQSENT
|
6.5 | IC50 | 2 | — |