Target Details
| UniProt AC | P03366 |
|---|---|
| Gene Symbol | gag-pol |
| Protein Name | Gag-Pol polyprotein |
| Organism | Human immunodeficiency virus type 1 group M subtype B (isolate BH10) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00540 (Gag_p17) PF19317 (Gag_p24_C) PF00552 (IN_DBD_C) PF02022 (Integrase_Zn) PF00075 (RNase_H) PF00665 (rve) PF00077 (RVP) PF00078 (RVT_1) PF06815 (RVT_connect) PF06817 (RVT_thumb) PF00098 (zf-CCHC) |
Summary
- Multi-target molecules 580
- Clinical molecules 0
- Avg pChEMBL 7.7
Top Co-occurrence Targets
- env 319 shared
- pol 259 shared
- reverse transcriptase 6 shared
- pol 1 shared
- DHODH 1 shared
Active Molecules (580)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ALUIKCFZMKVHTN
|
8.8 | IC50 | 2 | — | |
BDVZDHYAODJKQO
|
8.8 | IC50 | 2 | — | |
BGBAKULBBCPHEZ
|
8.8 | IC50 | 2 | — | |
DYJUNFLDNLNNKC
|
8.8 | IC50 | 2 | — | |
IDPPOMXSOMVURH
|
8.8 | IC50 | 2 | — | |
IGIISKXSSNGGSZ
|
8.8 | IC50 | 2 | — | |
KLBYEVXRLYVRSJ
|
8.8 | IC50 | 2 | — | |
LDMXXWBXVJBFHG
|
8.8 | IC50 | 2 | — | |
OMMIQIUADGJCCZ
|
8.8 | IC50 | 2 | — | |
OPSFIOYSJJIXAG
|
8.8 | IC50 | 2 | — | |
QLKUDQVPNKOAGG
|
8.8 | IC50 | 2 | — | |
QYKCEACKZWPLGG
|
8.8 | IC50 | 2 | — | |
SVYBUPDUPFYKBO
|
8.8 | IC50 | 2 | — | |
SYNWTXZEYAFEPL
|
8.8 | IC50 | 2 | — | |
TVSVXKFRQOASMA
|
8.8 | IC50 | 2 | — | |
UGABXFVGDVVJJJ
|
8.8 | IC50 | 2 | — | |
VGKXNGHFULVQQJ
|
8.8 | IC50 | 2 | — | |
XGHUOLJRIMAJGZ
|
8.8 | IC50 | 2 | — | |
XIEMATKZJAJQEG
|
8.8 | IC50 | 2 | — | |
ZKSVTAPAFZBEPN
|
8.8 | IC50 | 2 | — | |
ZNWRCFAAHQDGLA
|
8.8 | IC50 | 2 | — | |
HFRNUFDENULMJC
|
8.7 | IC50 | 2 | — | |
HPKVFXFYAXATBI
|
8.7 | IC50 | 2 | — | |
LVLGERXURTXXSL
|
8.7 | IC50 | 2 | — | |
MIKFGLKTLFPBRR
|
8.7 | IC50 | 2 | — | |
OXVLCRQAZMVBLP
|
8.7 | IC50 | 2 | — | |
RTAYASJKNZLYHO
|
8.7 | IC50 | 2 | — | |
UDPKVAHRPQZWAP
|
8.7 | IC50 | 2 | — | |
XGHUOLJRIMAJGZ
|
8.7 | IC50 | 2 | — | |
XYHQGLMTNIGUMH
|
8.7 | IC50 | 2 | — | |
DIYJTMKINSXCRR
|
8.7 | IC50 | 2 | — | |
PBLXLMRRRQEDTA
|
8.7 | IC50 | 2 | — | |
XAJYYDAEXGSPBU
|
8.7 | IC50 | 2 | — | |
YNHSZPGJMRDCFZ
|
8.7 | IC50 | 2 | — | |
ZIFLPSUVMSZPHJ
|
8.7 | IC50 | 2 | — | |
ASYHNPXMUNFZRC
|
8.7 | IC50 | 2 | — | |
AZPRETJPGHVWHH
|
8.7 | IC50 | 2 | — | |
CBRGCLQURKHNLV
|
8.7 | IC50 | 2 | — | |
DAEGPJVIJXEGIH
|
8.7 | IC50 | 2 | — | |
DMVYHYVKYGHCAQ
|
8.7 | IC50 | 2 | — | |
LHMLOBGVTWRTQY
|
8.7 | IC50 | 2 | — | |
MDLOQVRZURLPOD
|
8.7 | IC50 | 2 | — | |
NAJLYKFHDLKVPY
|
8.7 | IC50 | 2 | — | |
NRPIAQISVKJVKC
|
8.7 | IC50 | 2 | — | |
OXEKPZXYRYBHJX
|
8.7 | IC50 | 2 | — | |
PDYNCCKJYBGUQE
|
8.7 | IC50 | 2 | — | |
PZNXPIKYOCIJGV
|
8.7 | IC50 | 2 | — | |
QLVHHSZMLYWZLU
|
8.7 | IC50 | 2 | — | |
UGSNYSFOZKVFOB
|
8.7 | IC50 | 2 | — | |
VYLJLELAIADLHA
|
8.7 | IC50 | 2 | — |