Target Details
| UniProt AC | P02766 |
|---|---|
| Gene Symbol | TTR |
| Protein Name | Transthyretin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00576 (Transthyretin) |
Summary
- Multi-target molecules 125
- Clinical molecules 4
- Avg pChEMBL 7.33
KEGG Pathways (1)
Associated Diseases (3)
Active Molecules (125)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SIRUQHYFMOSYSV
|
7.0 | IC50 | 2 | — | |
RBQLXMYNDSQCDM
|
7.0 | IC50 | 2 | — | |
YMIKBDAUQJXFLA
|
7.0 | IC50 | 2 | — | |
FFWLYIPCGDWQBE
|
6.8 | IC50 | 2 | — | |
YEZNLOUZAIOMLT
|
6.8 | Kd | 3 | — | |
RMKSAIFOYKMQFY
|
6.8 | IC50 | 2 | — | |
GRRQKTDHGYEAAA
|
6.7 | IC50 | 2 | — | |
RPHMYDAWGOVIJU
|
6.7 | IC50 | 2 | — | |
WHQCHUCQKNIQEC
|
6.7 | Kd | 6 | — | |
DCOPUUMXTXDBNB
|
6.6 | Kd | 5 | — | |
SGHDFUMUJLRANA
|
6.6 | IC50 | 2 | — | |
ZOMDKNTVDCFYQX
|
6.6 | IC50 | 2 | — | |
FYQAHXWSEBYCMQ
|
6.5 | IC50 | 2 | — | |
JZFPYUNJRRFVQU
|
6.5 | IC50 | 2 | — | |
XRKNSSRFHTUUGW
|
6.4 | IC50 | 2 | — | |
HUPFGZXOMWLGNK
|
6.4 | Kd | 3 | Yes | |
LUKBXSAWLPMMSZ
|
6.3 | Kd | 18 | Yes | |
SBDNJUWAMKYJOX
|
6.3 | IC50 | 5 | — | |
AVALWFKKPLBJCO
|
6.3 | Kd | 2 | — | |
KZNIFHPLKGYRTM
|
6.2 | IC50 | 21 | Yes | |
FEXBXMFVRKZOOZ
|
6.2 | Kd | 2 | — | |
CVCXGSKKNFKCRH
|
6.1 | IC50 | 2 | — | |
NGJLOFCOEOHFKQ
|
6.1 | IC50 | 4 | — | |
UYJQGBUMNGFPIF
|
6.1 | IC50 | 2 | — | |
WMHVUSFNJBJQQB
|
6.1 | IC50 | 2 | — |