Target Details
| UniProt AC | P01130 |
|---|---|
| Gene Symbol | LDLR |
| Protein Name | Low-density lipoprotein receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07645 (EGF_CA) PF14670 (FXa_inhibition) PF00057 (Ldl_recept_a) PF00058 (Ldl_recept_b) |
Summary
- Multi-target molecules 224
- Clinical molecules 0
- Avg pChEMBL 6.85
KEGG Pathways (11)
Associated Diseases (4)
Active Molecules (224)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RXGJEHGKLXXJLS
|
6.3 | IC50 | 2 | — | |
SNBPWJVDOPZESG
|
6.3 | IC50 | 2 | — | |
TYAQBURXLGATKD
|
6.3 | IC50 | 2 | — | |
TYIYZRBWVAEQDY
|
6.3 | IC50 | 2 | — | |
ULJDGEPOAMADRJ
|
6.3 | IC50 | 2 | — | |
VGPQXXHISQYBNH
|
6.3 | IC50 | 2 | — | |
VNNSUPKAKVZRAS
|
6.3 | IC50 | 2 | — | |
WKJXNKGPJMUFPV
|
6.3 | IC50 | 2 | — | |
WVBBQINPROFUTD
|
6.3 | IC50 | 2 | — | |
XDEISTVXIHIEEY
|
6.3 | IC50 | 2 | — | |
XLZSMKCEQYOUBB
|
6.3 | IC50 | 2 | — | |
XSFJGBZVNFHACL
|
6.3 | IC50 | 2 | — | |
XSICDJDMSHRDIV
|
6.3 | IC50 | 2 | — | |
XXFKDDJGZGVTLW
|
6.3 | IC50 | 2 | — | |
XZABVPJOOVOYTI
|
6.3 | IC50 | 2 | — | |
ZFWIQMUIHYZSOF
|
6.3 | IC50 | 2 | — | |
VOAMXMMBZJDXSU
|
6.2 | Ki | 2 | — | |
NHJUFNWIIVOTIH
|
6.2 | IC50 | 2 | — | |
FPILCJQVCVIRHQ
|
6.2 | IC50 | 2 | — | |
AVCCKFHOOJRTCR
|
6.1 | IC50 | 2 | — | |
TYKXIBLBQNRTJM
|
6.1 | IC50 | 2 | — | |
ORPZALWAWWEEDP
|
6.1 | IC50 | 2 | — | |
GOXJDJCGIHVGAY
|
6.0 | Ki | 2 | — | |
SGJYNXWRJNILLN
|
6.0 | Ki | 2 | — |