Target Details
| UniProt AC | P01130 |
|---|---|
| Gene Symbol | LDLR |
| Protein Name | Low-density lipoprotein receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07645 (EGF_CA) PF14670 (FXa_inhibition) PF00057 (Ldl_recept_a) PF00058 (Ldl_recept_b) |
Summary
- Multi-target molecules 224
- Clinical molecules 0
- Avg pChEMBL 6.85
KEGG Pathways (11)
Associated Diseases (4)
Active Molecules (224)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WEBMSJYTWXDLIP
|
6.4 | IC50 | 2 | — | |
BJBASKROIULEMR
|
6.4 | Ki | 2 | — | |
FSWBQPGSMBLQBY
|
6.4 | IC50 | 2 | — | |
RIMRVERSFDYITK
|
6.3 | IC50 | 2 | — | |
WDOZXDCBSSIRIX
|
6.3 | Ki | 2 | — | |
SUNSLACFIOGRFF
|
6.3 | IC50 | 2 | — | |
ALPNZVCVPJFQIU
|
6.3 | IC50 | 2 | — | |
AZFPODXRUNPZHM
|
6.3 | IC50 | 2 | — | |
BOEQQAQLLWKPTJ
|
6.3 | IC50 | 2 | — | |
BRBNSXUDJYDTAG
|
6.3 | IC50 | 2 | — | |
BTAAQTWWDLUMTF
|
6.3 | IC50 | 2 | — | |
CNGCIJQYBFMRMX
|
6.3 | IC50 | 2 | — | |
CRYTZKVYOZQLRR
|
6.3 | IC50 | 2 | — | |
CUHBJMSOISXVMR
|
6.3 | IC50 | 2 | — | |
DCPMQDCTYSJULX
|
6.3 | IC50 | 2 | — | |
DNZWZESQXUDNMY
|
6.3 | IC50 | 2 | — | |
DONIEJUKPWBLFP
|
6.3 | IC50 | 2 | — | |
DSUVELDKXDKGHU
|
6.3 | IC50 | 2 | — | |
FMNPUNYDOXDGJL
|
6.3 | IC50 | 2 | — | |
FOZMZJIMMVCKDE
|
6.3 | IC50 | 2 | — | |
FTHXTCAXAGRYFO
|
6.3 | IC50 | 2 | — | |
GJJNMAVROKHYBE
|
6.3 | IC50 | 2 | — | |
GNZYKGNQNCDUGS
|
6.3 | IC50 | 2 | — | |
GYDLBEUNRPUORD
|
6.3 | IC50 | 2 | — | |
GYRYVQSHMAAQKC
|
6.3 | IC50 | 2 | — | |
HJJJHFVYQDSEFZ
|
6.3 | IC50 | 2 | — | |
HMSVYVLLKIGLFT
|
6.3 | IC50 | 2 | — | |
HVRHTDCRQSHYOI
|
6.3 | IC50 | 2 | — | |
IJMDXLMQQXPEEX
|
6.3 | IC50 | 2 | — | |
JGLBVZXAFLSBCU
|
6.3 | IC50 | 2 | — | |
JRGJGUZUUUKIDC
|
6.3 | IC50 | 2 | — | |
KASDPFCBFIWJGE
|
6.3 | IC50 | 2 | — | |
KYENQZFDWAELLQ
|
6.3 | IC50 | 2 | — | |
LQNHCVGOZPMYOV
|
6.3 | IC50 | 2 | — | |
LTZLQMSMMBBVJA
|
6.3 | IC50 | 2 | — | |
LYMYTGOIKDBELY
|
6.3 | IC50 | 2 | — | |
MOYBXIHKSBVEGD
|
6.3 | IC50 | 2 | — | |
NNDLHUHLCVZCQG
|
6.3 | IC50 | 2 | — | |
NXAWESRPHOWAJS
|
6.3 | IC50 | 2 | — | |
OKDDJQPOHMWTNM
|
6.3 | IC50 | 2 | — | |
ORVGAHROAPZBAA
|
6.3 | IC50 | 2 | — | |
OSLDLYWXYKWSBN
|
6.3 | IC50 | 2 | — | |
PBFLCRPIXMRFSM
|
6.3 | IC50 | 2 | — | |
PRCZAYMEHYDTNS
|
6.3 | IC50 | 2 | — | |
PRMMNARWNYGQRR
|
6.3 | IC50 | 2 | — | |
QBEFLWKVIFFKMQ
|
6.3 | IC50 | 2 | — | |
QFEZLQHDFGWYBB
|
6.3 | IC50 | 2 | — | |
QKHPCEZOONLJGL
|
6.3 | IC50 | 2 | — | |
QSQIUHYDUXLSSG
|
6.3 | IC50 | 2 | — | |
RDEQYXISVCQQMO
|
6.3 | IC50 | 2 | — |