Target Details
| UniProt AC | P01130 |
|---|---|
| Gene Symbol | LDLR |
| Protein Name | Low-density lipoprotein receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07645 (EGF_CA) PF14670 (FXa_inhibition) PF00057 (Ldl_recept_a) PF00058 (Ldl_recept_b) |
Summary
- Multi-target molecules 224
- Clinical molecules 0
- Avg pChEMBL 6.85
KEGG Pathways (11)
Associated Diseases (4)
Active Molecules (224)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DQUNQCNBDRFHIT
|
6.9 | IC50 | 2 | — | |
GLLGKKKZWFJJCJ
|
6.9 | IC50 | 2 | — | |
KHEZVUTYPQPKMX
|
6.9 | IC50 | 2 | — | |
QKZPDRYLXKUIDB
|
6.9 | IC50 | 2 | — | |
QWSRELJSYBDPRL
|
6.9 | IC50 | 2 | — | |
RMKDHFDRCBWRPZ
|
6.9 | IC50 | 2 | — | |
WNRKBYIGXJGAEI
|
6.9 | IC50 | 2 | — | |
XLEYVMNOFVCPKK
|
6.9 | IC50 | 2 | — | |
IIACQYHQRJCFAR
|
6.9 | IC50 | 2 | — | |
VZNVNRHFHPQHQA
|
6.9 | Ki | 2 | — | |
AAYMIURIOIEXPG
|
6.8 | IC50 | 2 | — | |
AMADQZYKECSVOD
|
6.8 | IC50 | 2 | — | |
AROYUBVLQGLEJW
|
6.8 | IC50 | 2 | — | |
BCVVUQJCTFVPPX
|
6.8 | IC50 | 2 | — | |
BJVXVQYMRIDQSO
|
6.8 | IC50 | 2 | — | |
BKNYGFCMSQXXAY
|
6.8 | IC50 | 2 | — | |
CIAMVYSKSRDHKW
|
6.8 | IC50 | 2 | — | |
DCIMYVGIHVXZCW
|
6.8 | IC50 | 2 | — | |
DPSAHQIWNWXORF
|
6.8 | IC50 | 2 | — | |
FGKBFNJXPBUFBF
|
6.8 | IC50 | 2 | — | |
FHQIQLZORIIJCJ
|
6.8 | IC50 | 2 | — | |
GBYGLFAUNQRUSD
|
6.8 | IC50 | 2 | — | |
GCTYLQDZFAOXNZ
|
6.8 | IC50 | 2 | — | |
HSOKWOADSAANKP
|
6.8 | IC50 | 2 | — | |
IVPXAHSPNMQFGV
|
6.8 | IC50 | 2 | — | |
LCYSOOPHKDMGSN
|
6.8 | IC50 | 2 | — | |
LPZRZOQXPIDWJC
|
6.8 | IC50 | 2 | — | |
MDOITGFKFKPKCN
|
6.8 | IC50 | 2 | — | |
MYGQCSYJOCJPFB
|
6.8 | IC50 | 2 | — | |
MZWCZQFAKFQXAQ
|
6.8 | IC50 | 2 | — | |
NBBMJWKHBJDFGL
|
6.8 | IC50 | 2 | — | |
NNXNKSOVYSLSFY
|
6.8 | IC50 | 2 | — | |
PFISJUXNQBLIRP
|
6.8 | IC50 | 2 | — | |
PJHDLPARKAVICN
|
6.8 | IC50 | 2 | — | |
QBMRJRDZKQIKCP
|
6.8 | IC50 | 2 | — | |
QHFAKOAIOHFGAG
|
6.8 | IC50 | 2 | — | |
ROCUVPFOJQUBBQ
|
6.8 | IC50 | 2 | — | |
SCMDQZAAPDKIHV
|
6.8 | IC50 | 2 | — | |
UUXNLVNUARUQPI
|
6.8 | IC50 | 2 | — | |
VGAZTZLZPGZMAZ
|
6.8 | IC50 | 2 | — | |
VQEZXIWIQYERPR
|
6.8 | IC50 | 2 | — | |
VXNVOKZEOXXHKP
|
6.8 | IC50 | 2 | — | |
WCLSBIUNDNBREO
|
6.8 | IC50 | 2 | — | |
YCVOWOOAPJRRBI
|
6.8 | IC50 | 2 | — | |
ZMDVAPWVJYZESL
|
6.8 | IC50 | 2 | — | |
ZYRHDMLWKCRPIC
|
6.7 | Ki | 2 | — | |
JUMIZFILSSYEFV
|
6.6 | Ki | 2 | — | |
XRPADFDSTLJKJR
|
6.5 | Ki | 2 | — | |
FRMJPXCBCWOLHG
|
6.4 | Ki | 2 | — | |
VVFBDPKAWCMBFC
|
6.4 | IC50 | 2 | — |