Target Details
| UniProt AC | P01130 |
|---|---|
| Gene Symbol | LDLR |
| Protein Name | Low-density lipoprotein receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07645 (EGF_CA) PF14670 (FXa_inhibition) PF00057 (Ldl_recept_a) PF00058 (Ldl_recept_b) |
Summary
- Multi-target molecules 224
- Clinical molecules 0
- Avg pChEMBL 6.85
KEGG Pathways (11)
Associated Diseases (4)
Active Molecules (224)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OHMWYKRRPHNKAY
|
7.3 | IC50 | 2 | — | |
OOBXOHWMTQHGPZ
|
7.3 | IC50 | 2 | — | |
OTAKLFUVEQRFQC
|
7.3 | IC50 | 2 | — | |
OUHIHZKBZJHMKN
|
7.3 | IC50 | 2 | — | |
OUHIHZKBZJHMKN
|
7.3 | IC50 | 2 | — | |
PEFANKFLDJZTTE
|
7.3 | IC50 | 2 | — | |
PKLWPELHYNFFSC
|
7.3 | IC50 | 2 | — | |
PMMGPFKPCNXWKH
|
7.3 | IC50 | 2 | — | |
PQCJVPLQTYCXHG
|
7.3 | IC50 | 2 | — | |
PSNROLOZFCGPOO
|
7.3 | IC50 | 2 | — | |
QRIOCRNXOURWNI
|
7.3 | IC50 | 2 | — | |
RBWKHLPGHMYEBU
|
7.3 | IC50 | 2 | — | |
RZFKCVRKHPUZSA
|
7.3 | IC50 | 2 | — | |
SIUIJEXTVIHXRM
|
7.3 | IC50 | 2 | — | |
SREPCAPKCNETHI
|
7.3 | IC50 | 2 | — | |
SROMRSNBDIXBNC
|
7.3 | IC50 | 2 | — | |
SZGNJXJONFTTMZ
|
7.3 | IC50 | 2 | — | |
TVWRUGYHFKQXJI
|
7.3 | IC50 | 2 | — | |
UPZHBFNFWJCORK
|
7.3 | IC50 | 2 | — | |
UTOIMUBAPYEYBD
|
7.3 | IC50 | 2 | — | |
UTPUESWLNFEKOJ
|
7.3 | IC50 | 2 | — | |
UYTBZWJKJSZDPS
|
7.3 | IC50 | 2 | — | |
VEBUCFXLBZQBKJ
|
7.3 | IC50 | 2 | — | |
VEEBNTLUXIEQDX
|
7.3 | IC50 | 2 | — | |
VEJNOLOAWWWCED
|
7.3 | IC50 | 2 | — | |
WBHDYRHQHHLKQI
|
7.3 | IC50 | 2 | — | |
WKKAQOPQRBMISJ
|
7.3 | IC50 | 2 | — | |
WRPFBABRQIASOS
|
7.3 | IC50 | 2 | — | |
XBMWLWQWZMXFJE
|
7.3 | IC50 | 2 | — | |
XCIVVNWSQRGLMD
|
7.3 | IC50 | 2 | — | |
XJIUUGQYWJGRIR
|
7.3 | IC50 | 2 | — | |
XODWNXFGTNVYHB
|
7.3 | IC50 | 2 | — | |
XUATYLDPLNNZEX
|
7.3 | IC50 | 2 | — | |
YFTHABGMWCGOAK
|
7.3 | IC50 | 2 | — | |
ZDFSJIHCRYLAMT
|
7.3 | IC50 | 2 | — | |
ZQFZHVFJXFINPM
|
7.3 | IC50 | 2 | — | |
ZWPQEWXCTYEVJU
|
7.3 | IC50 | 2 | — | |
HGLMFBHBAMWYHY
|
7.2 | Ki | 2 | — | |
NSTFRFKCUDSCEN
|
7.2 | Ki | 2 | — | |
AFTCBZMZKYOMRS
|
7.1 | IC50 | 3 | — | |
OTKKOUJLPCKSCD
|
7.1 | Ki | 2 | — | |
XZNCSFCXWWVUCW
|
7.0 | Ki | 2 | — | |
OMZKYRSDRNYKAZ
|
7.0 | Ki | 2 | — | |
PINVMNVLSVYQKP
|
7.0 | Ki | 2 | — | |
KLPYFSFJVFMBJS
|
7.0 | Ki | 2 | — | |
VORHKYQSFSQEEO
|
7.0 | Ki | 2 | — | |
SXUMLHZCSVRHKE
|
6.9 | IC50 | 2 | — | |
BDEUYEAHVFTURG
|
6.9 | IC50 | 2 | — | |
BEILGIKXQDGLEW
|
6.9 | IC50 | 2 | — | |
CTWNVUQVDCMLSE
|
6.9 | IC50 | 2 | — |