Target Details
UniProt ACP01130
Gene SymbolLDLR
Protein NameLow-density lipoprotein receptor
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF07645 (EGF_CA) PF14670 (FXa_inhibition) PF00057 (Ldl_recept_a) PF00058 (Ldl_recept_b)
Summary
  • Multi-target molecules 224
  • Clinical molecules 0
  • Avg pChEMBL 6.85
Top Co-occurrence Targets
Active Molecules (224)
InChIKey pChEMBL Type Targets Clinical
KKTRCZWTWYYSCY 8.7 IC50 2
AJCMEMYQDXJTLA 8.5 IC50 2
PYVKCKXGZHKWHI 8.2 IC50 2
PNXFQQVLICCBOG 8.1 IC50 2
MVKQIKVUJHXYFL 7.8 Ki 2
MUNCMINBJLDFBS 7.8 Ki 2
PGYQBTHDSQHEAE 7.6 Ki 2
GEYNSTBJBJHKBR 7.6 Ki 2
ZRUWDDBTCYFPLA 7.6 Ki 2
CXYIZMOWQIOCCP 7.4 Ki 2
WRHMMJSLZQKTIJ 7.3 Ki 2
TZQCDWGPFXCCFJ 7.3 Ki 2
ASTBLTXEDYOOHH 7.3 IC50 2
BFBKGIZCMYXWKP 7.3 IC50 2
BPABXCYDPRUTJP 7.3 IC50 2
BPDDXYVTWKHSPJ 7.3 IC50 2
BYCVINHSHUVRLH 7.3 IC50 2
CBNRIGHHWFOMTR 7.3 IC50 2
CMEDPZMTGNTTBQ 7.3 IC50 2
DAFOIRPOHRTCCU 7.3 IC50 2
DQNPOFYOPIYJIW 7.3 IC50 2
FAQXSFYHHVOERA 7.3 IC50 2
FIGHUWBUPINGCK 7.3 IC50 2
FIGQUGWNWAGSMX 7.3 IC50 2
FVSGRCFFDUJBSM 7.3 IC50 2
GHYVELVQBCQZAW 7.3 IC50 2
HJWRADTVRMRTCL 7.3 IC50 2
HSGRVVJDCMQDDO 7.3 IC50 2
HSVBNERTWMNCEC 7.3 IC50 2
HTZAUHJLSZVMER 7.3 IC50 2
HVQDJWFAGPSFHW 7.3 IC50 2
HZSDNSSEFWHOAM 7.3 IC50 2
IBHCNYFVFVJSNW 7.3 IC50 2
IMEFOOHITUHVKM 7.3 IC50 2
IOHQDPRJGZKIKP 7.3 IC50 2
ISQOVBPPZKQLLB 7.3 IC50 2
IVTNLJRCNTZRGT 7.3 IC50 2
JBUXHFKZMXLWCD 7.3 IC50 2
JGLBVZXAFLSBCU 7.3 IC50 2
JHYDAIUPBQLKHW 7.3 IC50 2
JQXBYNLOSRYECM 7.3 IC50 2
KDFJEZBQMMRKJX 7.3 IC50 2
KICTXGZKQYJVHU 7.3 IC50 2
KJNMWJFZUNTGKI 7.3 IC50 2
LBFGAFNKUVYELA 7.3 IC50 2
LPLOQDKAJJIQHJ 7.3 IC50 2
MFZAHCDUXVQHDG 7.3 IC50 2
NHAKTDNLCUBYIO 7.3 IC50 2
NRRUCUBIKFVVTF 7.3 IC50 2
NRZSNKPBLRFRCO 7.3 IC50 2
2D structure