Target Details
| UniProt AC | P01130 |
|---|---|
| Gene Symbol | LDLR |
| Protein Name | Low-density lipoprotein receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07645 (EGF_CA) PF14670 (FXa_inhibition) PF00057 (Ldl_recept_a) PF00058 (Ldl_recept_b) |
Summary
- Multi-target molecules 224
- Clinical molecules 0
- Avg pChEMBL 6.85
KEGG Pathways (11)
Associated Diseases (4)
Active Molecules (224)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KKTRCZWTWYYSCY
|
8.7 | IC50 | 2 | — | |
AJCMEMYQDXJTLA
|
8.5 | IC50 | 2 | — | |
PYVKCKXGZHKWHI
|
8.2 | IC50 | 2 | — | |
PNXFQQVLICCBOG
|
8.1 | IC50 | 2 | — | |
MVKQIKVUJHXYFL
|
7.8 | Ki | 2 | — | |
MUNCMINBJLDFBS
|
7.8 | Ki | 2 | — | |
PGYQBTHDSQHEAE
|
7.6 | Ki | 2 | — | |
GEYNSTBJBJHKBR
|
7.6 | Ki | 2 | — | |
ZRUWDDBTCYFPLA
|
7.6 | Ki | 2 | — | |
CXYIZMOWQIOCCP
|
7.4 | Ki | 2 | — | |
WRHMMJSLZQKTIJ
|
7.3 | Ki | 2 | — | |
TZQCDWGPFXCCFJ
|
7.3 | Ki | 2 | — | |
ASTBLTXEDYOOHH
|
7.3 | IC50 | 2 | — | |
BFBKGIZCMYXWKP
|
7.3 | IC50 | 2 | — | |
BPABXCYDPRUTJP
|
7.3 | IC50 | 2 | — | |
BPDDXYVTWKHSPJ
|
7.3 | IC50 | 2 | — | |
BYCVINHSHUVRLH
|
7.3 | IC50 | 2 | — | |
CBNRIGHHWFOMTR
|
7.3 | IC50 | 2 | — | |
CMEDPZMTGNTTBQ
|
7.3 | IC50 | 2 | — | |
DAFOIRPOHRTCCU
|
7.3 | IC50 | 2 | — | |
DQNPOFYOPIYJIW
|
7.3 | IC50 | 2 | — | |
FAQXSFYHHVOERA
|
7.3 | IC50 | 2 | — | |
FIGHUWBUPINGCK
|
7.3 | IC50 | 2 | — | |
FIGQUGWNWAGSMX
|
7.3 | IC50 | 2 | — | |
FVSGRCFFDUJBSM
|
7.3 | IC50 | 2 | — | |
GHYVELVQBCQZAW
|
7.3 | IC50 | 2 | — | |
HJWRADTVRMRTCL
|
7.3 | IC50 | 2 | — | |
HSGRVVJDCMQDDO
|
7.3 | IC50 | 2 | — | |
HSVBNERTWMNCEC
|
7.3 | IC50 | 2 | — | |
HTZAUHJLSZVMER
|
7.3 | IC50 | 2 | — | |
HVQDJWFAGPSFHW
|
7.3 | IC50 | 2 | — | |
HZSDNSSEFWHOAM
|
7.3 | IC50 | 2 | — | |
IBHCNYFVFVJSNW
|
7.3 | IC50 | 2 | — | |
IMEFOOHITUHVKM
|
7.3 | IC50 | 2 | — | |
IOHQDPRJGZKIKP
|
7.3 | IC50 | 2 | — | |
ISQOVBPPZKQLLB
|
7.3 | IC50 | 2 | — | |
IVTNLJRCNTZRGT
|
7.3 | IC50 | 2 | — | |
JBUXHFKZMXLWCD
|
7.3 | IC50 | 2 | — | |
JGLBVZXAFLSBCU
|
7.3 | IC50 | 2 | — | |
JHYDAIUPBQLKHW
|
7.3 | IC50 | 2 | — | |
JQXBYNLOSRYECM
|
7.3 | IC50 | 2 | — | |
KDFJEZBQMMRKJX
|
7.3 | IC50 | 2 | — | |
KICTXGZKQYJVHU
|
7.3 | IC50 | 2 | — | |
KJNMWJFZUNTGKI
|
7.3 | IC50 | 2 | — | |
LBFGAFNKUVYELA
|
7.3 | IC50 | 2 | — | |
LPLOQDKAJJIQHJ
|
7.3 | IC50 | 2 | — | |
MFZAHCDUXVQHDG
|
7.3 | IC50 | 2 | — | |
NHAKTDNLCUBYIO
|
7.3 | IC50 | 2 | — | |
NRRUCUBIKFVVTF
|
7.3 | IC50 | 2 | — | |
NRZSNKPBLRFRCO
|
7.3 | IC50 | 2 | — |