Target Details
| UniProt AC | P01127 |
|---|---|
| Gene Symbol | PDGFB |
| Protein Name | Platelet-derived growth factor subunit B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00341 (PDGF) PF04692 (PDGF_N) |
Summary
- Multi-target molecules 16
- Clinical molecules 0
- Avg pChEMBL 7.47
KEGG Pathways (21)
- Calcium signaling pathway
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- Fluid shear stress and atherosclerosis
- Focal adhesion
- Gap junction
- Glioma
- Integrin signaling
- JAK-STAT signaling pathway
- Kaposi sarcoma-associated herpesvirus infection
- MAPK signaling pathway
- Melanoma
- MicroRNAs in cancer
- PI3K-Akt signaling pathway
- Pathways in cancer
- Phospholipase D signaling pathway
- Prostate cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Renal cell carcinoma
Associated Diseases (4)
Active Molecules (16)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JWITUUPNOFPOGN
|
8.0 | IC50 | 3 | — | |
JZKVGXOGXXCAKW
|
8.0 | IC50 | 3 | — | |
DQGTWWTUKZRUKI
|
8.0 | IC50 | 3 | — | |
KESUAIOCJKBPRI
|
7.9 | IC50 | 3 | — | |
ZLUSJKSRLQNGJZ
|
7.8 | IC50 | 3 | — | |
QEUJPSURIIRPKP
|
7.8 | IC50 | 3 | — | |
IJAYHJGVTCMSHM
|
7.7 | IC50 | 3 | — | |
HIQVRUAZLKNDKM
|
7.7 | IC50 | 3 | — | |
GESXFTKSUVVIGO
|
7.6 | IC50 | 3 | — | |
KWCIURFGWLVSPG
|
7.5 | IC50 | 3 | — | |
YXOIGKRFYLDKCK
|
7.3 | IC50 | 3 | — | |
YRGIFNDOEPYLFQ
|
6.9 | IC50 | 3 | — | |
OJFKUJDRGJSAQB
|
6.9 | IC50 | 17 | — | |
LVCMBVIHFUNWCJ
|
6.8 | IC50 | 3 | — | |
SOBFCBCYWSMQOU
|
6.8 | IC50 | 3 | — | |
YDTJZVVELNGMQL
|
6.6 | IC50 | 3 | — |