Target Details
| UniProt AC | P00808 |
|---|---|
| Gene Symbol | penP |
| Protein Name | Beta-lactamase |
| Organism | Bacillus licheniformis |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13354 (Beta-lactamase2) |
Summary
- Multi-target molecules 2
- Clinical molecules 0
- Avg pChEMBL 6.39
Top Co-occurrence Targets
- OXA-1 2 shared
- blaZ 2 shared
- KPC-2 1 shared
- blaUOE-1 1 shared
- bla OXY 1 shared
- blaTEM-1 1 shared
- blaTEM-125 1 shared
- 1 shared
- imiA 1 shared
- blaCTX-M-53 1 shared
Active Molecules (2)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JYGFUXUBGZBBAC
|
6.5 | IC50 | 5 | — | |
LPQZKKCYTLCDGQ
|
6.3 | IC50 | 15 | — |