Target Details
| UniProt AC | P00800 |
|---|---|
| Gene Symbol | npr |
| Protein Name | Thermolysin |
| Organism | Bacillus thermoproteolyticus |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF07504 (FTP) PF03413 (PepSY) PF01447 (Peptidase_M4) PF02868 (Peptidase_M4_C) |
Summary
- Multi-target molecules 12
- Clinical molecules 0
- Avg pChEMBL 7.82
Active Molecules (12)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MSUGUYPTEWUYIP
|
8.7 | IC50 | 2 | — | |
OJCFZTVYDSKXNM
|
8.5 | IC50 | 4 | — | |
OJCFZTVYDSKXNM
|
8.5 | IC50 | 5 | — | |
MIQFXJKPZRPRNQ
|
8.3 | IC50 | 2 | — | |
VFEZBZKVMQPXIZ
|
8.3 | IC50 | 2 | — | |
VUEMZVPEAVUVHY
|
8.2 | IC50 | 2 | — | |
FBJRJRIBPSETON
|
8.1 | IC50 | 2 | — | |
ZPHBZEQOLSRPAK
|
7.5 | Ki | 2 | — | |
ZPHBZEQOLSRPAK
|
7.5 | IC50 | 5 | — | |
MCEAHFJYQBFRCJ
|
7.2 | IC50 | 2 | — | |
FGSNBBSHVNLDMX
|
6.8 | IC50 | 2 | — | |
SZYXPUAQRACFJD
|
6.2 | IC50 | 2 | — |