Target Details
UniProt ACP00750
Gene SymbolPLAT
Protein NameTissue-type plasminogen activator
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00008 (EGF) PF00039 (fn1) PF00051 (Kringle) PF00089 (Trypsin)
Summary
  • Multi-target molecules 95
  • Clinical molecules 4
  • Avg pChEMBL 6.78
Top Co-occurrence Targets
Active Molecules (95)
InChIKey pChEMBL Type Targets Clinical
VCVSFHZQGWZRGK 6.5 IC50 4
RSJYFASOCLFHRR 6.5 Ki 6
BZGZTAKGLPGMAV 6.5 IC50 4
AACVRGGQVLDYDM 6.5 Ki 4
NKADRYHVDUCFQU 6.5 Ki 4
LTXLJGIDFWWEQI 6.4 Ki 4
QZIXPYQULZYTPK 6.4 Ki 2
YBSXFYTXULBNOE 6.4 Ki 6
BIHPYGVYKSQDLA 6.4 Ki 6
BVTBOJXEAPSOEB 6.3 Ki 6
IBHLYVDUKHZEBW 6.3 IC50 2
DCUODGWOKBGFJV 6.3 Ki 3
PKASBNFVFWUNOA 6.3 IC50 4
WQDOEYAJPUSQCH 6.3 IC50 6 Yes
DSEQCUGXKCOSSU 6.3 IC50 5
AJKIEWKQNYUUAZ 6.2 Ki 2
CFSQPEBVGUSQII 6.2 Ki 5
JSPAUBUYPPZXSG 6.2 Ki 17 Yes
LYVSCNRRXJZCRV 6.2 Ki 2
CQQFREVZNRVIIM 6.2 IC50 4
YLSKCQOVDOZHTQ 6.2 Ki 2
CSWQJKHBMACTGB 6.2 Ki 6
FVEMXCSGNPVPIT 6.2 Ki 4
BOMLKKNGTDVLHA 6.2 Ki 6
GJKMIUMNDMWVGF 6.2 IC50 5
WCFWDBPDMBXMTQ 6.2 Ki 3
LCSPIPBAMWVNCU 6.1 IC50 3
QFBJYRZRHFZHEL 6.1 Ki 4
JENOLOFVMYLCBZ 6.1 IC50 4
DXFJLEXWZBCHSJ 6.1 Ki 3
JRJYGGVSLMZUHU 6.1 IC50 3
LMGQGPVCSYOMNS 6.1 Ki 6
MMMVHDBARFPCLX 6.1 Ki 6
VYJOAYZRCNHDNG 6.1 Ki 6
GKFHRQMCFNIZHA 6.1 Ki 4
QNUYHZAYXDMWMT 6.1 IC50 5
CDJBWPMAVJSWPS 6.1 Ki 6
UTYMFQPKWLTXJA 6.1 Ki 3
DKWNMCUOEDMMIN 6.0 Ki 6
PUSXAFWVXFYXRA 6.0 IC50 2
JDXUSWQJCGTBLN 6.0 IC50 4
QWTIOQGNSLCKBH 6.0 IC50 3
FKTVUGSKIYLIGS 6.0 Ki 2
HSHVHNIOQTZSOQ 6.0 Ki 5
KWZZDFIUKWTKDC 6.0 Ki 3
2D structure