Target Details
UniProt ACP00750
Gene SymbolPLAT
Protein NameTissue-type plasminogen activator
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00008 (EGF) PF00039 (fn1) PF00051 (Kringle) PF00089 (Trypsin)
Summary
  • Multi-target molecules 95
  • Clinical molecules 4
  • Avg pChEMBL 6.78
Top Co-occurrence Targets
Active Molecules (95)
InChIKey pChEMBL Type Targets Clinical
KBJGRHGRZYRRHG 9.5 Ki 6
IHBRTJZRICMSLW 9.2 IC50 4
MZFNXDNNMBIFKH 9.2 IC50 3
PWVZGBVCDDZZNQ 8.5 Ki 3
FXFYPTZERULUBS 8.2 Ki 5
BKMLZHDSJSJXNS 8.2 Ki 3
DCUODGWOKBGFJV 8.2 Ki 3
QBRUSDXUXPAOCZ 8.0 IC50 2
VGQFBYXDHFTAHX 7.7 Ki 6
UNYWSFMNRIYRDN 7.7 Ki 3
VCTXERTXMIFGOA 7.7 IC50 2
HEARWCQIVJNHBP 7.5 IC50 4
WOLHGVQMGPTOEN 7.5 IC50 4
KAGLWQUWUNBAOO 7.5 IC50 5
NZEAENHOWXTKPM 7.5 IC50 5
GAVRMVQHHVMXFD 7.5 Ki 11
ZLSGXUVBYIIXKU 7.5 Ki 5
HECONMODEBIAKY 7.3 IC50 9
KZVJNASRNCDNTJ 7.3 Ki 4
UNIOGIZCWAGOKV 7.2 Ki 6
BUGKCANFLDYYKD 7.2 IC50 6
RHEKWNPDSIWZKZ 7.0 IC50 8
WQVBAYOMZJYFJK 7.0 IC50 8
MJPRZTFMWHJGMK 7.0 IC50 6 Yes
SJOGQFLRNCUNDK 7.0 Ki 5
ZKPKJBOKOMILAA 7.0 Ki 6
ANKIJLVYTUKGJM 7.0 Ki 6
NTNRVRBIIZBTBR 7.0 IC50 8
BRZYOTMFHLERHD 7.0 Ki 17 Yes
ALBWLRSLXFJFTE 7.0 Ki 5
FEKRWNWZMOSVBX 7.0 Ki 6
PFCOFKBCTGBATD 7.0 Ki 6
BIHPYGVYKSQDLA 7.0 Ki 5
HNGQAWXKSWVXIP 6.9 Ki 2
CROZVKXDALXCPS 6.9 IC50 6
HLWKBMWAJJZWIT 6.9 Ki 5
CDJAIRYCIJZATA 6.8 Ki 6
CVLTYFQCFUHCBP 6.8 IC50 5
SFGQHQOPLLWNCX 6.8 Ki 3
QHOGUHKKMFDODA 6.8 Ki 6
OVQWFZKRHDTPOD 6.8 IC50 7
QJVPWUIKUDMGJM 6.8 Ki 6
ZDMYKWNIEWNTLR 6.7 IC50 5
QRPASZARTYLGAR 6.7 Ki 2
JECHDKUWRBFZLB 6.6 Ki 5
KEWCBOBJEQHYIV 6.6 Ki 6
GOERAAJVARXHDP 6.6 IC50 4
BXSDRFZOPSIGSI 6.5 IC50 4
NZEDSGTYZINZBH 6.5 Ki 3
RUJOXQDERXMGDN 6.5 Ki 3
2D structure