Target Details
UniProt ACP00749
Gene SymbolPLAU
Protein NameUrokinase-type plasminogen activator
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00051 (Kringle) PF00089 (Trypsin)
Summary
  • Multi-target molecules 256
  • Clinical molecules 4
  • Avg pChEMBL 6.99
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (256)
InChIKey pChEMBL Type Targets Clinical
UIEFTXMHYNHGEZ 6.3 Ki 2
ADJQHSQKTGJTKA 6.3 Ki 3
JZMPKIDYZMZCPR 6.3 Ki 2
RUJOXQDERXMGDN 6.3 Ki 3
BRZYOTMFHLERHD 6.3 Ki 17 Yes
LYTDWOOGBXMQGQ 6.3 Ki 3
RPMUVLQJQRPMOJ 6.3 Ki 3
ADSBUUURIYITQD 6.3 Ki 3
CQQFREVZNRVIIM 6.3 IC50 4
QPBFLOWZPFHTHE 6.3 Ki 6
RMJHMNZGTJDKCS 6.3 IC50 4
CHAKXPPMMOYNDT 6.3 Ki 3
MEKFQRDWXPJRHC 6.3 Ki 2
PJDBBQFSBXNSTE 6.3 Ki 2
ZKCSMEOONDAYCX 6.3 Ki 2
NTUOVTZYWIFOND 6.2 Ki 2
FKUAJSCZSYQJSF 6.2 Ki 4
IRTLDLFAEDDTRD 6.2 Ki 3
ISIVCLJSXCJXFI 6.2 Ki 2
WQDOEYAJPUSQCH 6.2 IC50 6 Yes
YCEDGYUKLCNMJH 6.2 Ki 2
BZWGGDJFDXDKDF 6.2 Ki 2
DGCKICNEBFFWGE 6.2 IC50 4
PDOPCKAPHCDUPT 6.2 Ki 3
VICVHWDAOZFSIP 6.2 Ki 2
AECPTICWHONWNW 6.2 Ki 2
QUNDYCNUUZNGBN 6.2 Ki 2
WATXEHGLYJKXOF 6.2 Ki 3
FLCRMGKKLKMMAE 6.2 Ki 2
QGLTXLFHFVMPJH 6.1 Ki 3
SJMNJNRKVVVGRB 6.1 Ki 2
URJKRCBBKTXOHS 6.1 Ki 3
CFIDHIDGDXATPD 6.1 IC50 4
IOTRRXDZDXKPBV 6.1 Ki 2
BBSZLQMSIMSHSW 6.1 Ki 2
CPIYDJBFUUZJPG 6.1 Ki 4
IUZFOKCCMJNLLQ 6.1 Ki 2
QHYGSRQJBXWIGI 6.1 Ki 2
UTQHUKDNPXJOJT 6.1 Ki 3
VBGMRZGJUPHRLG 6.1 Ki 2
DDPUNJKAKZZDPA 6.1 Ki 2
IVGMDANEFALECQ 6.1 IC50 5
XJUKHMPGPODLSN 6.1 Ki 3
ZGIWEZAHQKLMLT 6.1 IC50 2
IDRHKJAGRANANS 6.1 Ki 2
JPGNPKIYCTXJPG 6.1 Ki 2
JZSOCPVJALRMLO 6.1 IC50 2
KFBQPRUUOPSVGX 6.1 Ki 3
LDVXQIPCZWWFLR 6.1 Ki 3
MWBNFSUYTZMPST 6.0 IC50 3
2D structure