Target Details
UniProt ACP00749
Gene SymbolPLAU
Protein NameUrokinase-type plasminogen activator
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00051 (Kringle) PF00089 (Trypsin)
Summary
  • Multi-target molecules 256
  • Clinical molecules 4
  • Avg pChEMBL 6.99
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (256)
InChIKey pChEMBL Type Targets Clinical
ZNNRUQNYKOFUES 6.7 Ki 2
IEKKKOCYKOJJBP 6.7 Ki 3
HSHVHNIOQTZSOQ 6.6 Ki 5
OLHRAPVKZSUQLY 6.6 Ki 2
PKASBNFVFWUNOA 6.6 IC50 4
TXSJYFVZTQULMK 6.6 Ki 2
WTZSIVZMLBYQIH 6.6 Ki 2
YDLRKIGZKOOXGX 6.6 Ki 3
GKEDWEKWBQHEDD 6.6 Ki 3
YERQOXAYAFWFEJ 6.6 Ki 2
FZFPHLPTMPLMFJ 6.6 IC50 2
UVAYEBNBNNJWHZ 6.6 Ki 3
GDPHNLIBJUAUNC 6.6 Ki 3
IHVADESBZZCEJN 6.6 Ki 2
OPAXFTFGGLWWEL 6.6 Ki 2
UDURDZYWNVFIOM 6.6 Ki 4
DMRSHSWYVATHJS 6.6 Ki 2
CVKDCLNWMMYRKW 6.5 Ki 2
NDTNHGKZDUSWEQ 6.5 Ki 4
XKCHOMIJYLHXLI 6.5 Ki 2
YCMUIWWODVYRLS 6.5 Ki 3
FAKOUAJYWRNFEF 6.5 Ki 3
ABVQGTJUWOIMBS 6.5 Ki 2
ANMPAJKPHPHBMW 6.5 Ki 2
NFJBOMRZPXKWOS 6.5 Ki 3
ZOKSKHWGOAWJSA 6.5 IC50 4
VKFGNQCXLCROIA 6.5 Ki 4
ZGTBPFPYIIGPEC 6.5 Ki 4
FLKQFRKNGNJBNP 6.5 Ki 2
IXSDUZZGDXIMDY 6.5 Ki 3
OZCONSDLQBPMQO 6.5 Ki 2
JBMZFGZQZPOAGJ 6.5 Ki 3
MJPRZTFMWHJGMK 6.5 IC50 6 Yes
AKKWRLYFNUWVJB 6.5 Ki 4
RHERGFOYZXTLSI 6.5 Ki 3
FSCCYDSFQBJKGI 6.4 Ki 2
FHSUBJCOLTZQHR 6.4 Ki 3
FKTVUGSKIYLIGS 6.4 Ki 2
ICGQEIJGXOAEKE 6.4 Ki 3
KXSZMPGKDDBJRE 6.4 IC50 3
LMGQGPVCSYOMNS 6.4 Ki 6
AJKIEWKQNYUUAZ 6.4 Ki 2
ISJSHQTWOHGCMM 6.4 Ki 5
YKGYIDJEEQRWQH 6.4 IC50 6
ZSGVNBVMZBRWIM 6.4 Ki 3
OGMFURJUWYVEFV 6.4 Ki 2
WQDQVYGCTAVNKI 6.4 IC50 3
DMULMZBZVBBWBY 6.3 Ki 2
JXOUQPJAWDJHOP 6.3 Ki 2
SIYHDAGPPJTNHW 6.3 IC50 4
2D structure