Target Details
UniProt ACP00749
Gene SymbolPLAU
Protein NameUrokinase-type plasminogen activator
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00051 (Kringle) PF00089 (Trypsin)
Summary
  • Multi-target molecules 256
  • Clinical molecules 4
  • Avg pChEMBL 6.99
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (256)
InChIKey pChEMBL Type Targets Clinical
QJVPWUIKUDMGJM 7.0 Ki 6
VLUCTQXBQVXUNP 7.0 Ki 2
HZNLMAXGKJQXSL 7.0 Ki 2
BOMLKKNGTDVLHA 7.0 Ki 6
QRPASZARTYLGAR 7.0 Ki 2
OMMIMDGHTTXEFT 7.0 Ki 2
CDJBWPMAVJSWPS 7.0 Ki 6
ALBWLRSLXFJFTE 7.0 Ki 5
ZKQPJCFASKEYAL 7.0 Ki 2
HFUGBKCICWUZIJ 6.9 Ki 3
GDNFCRISLXZPOR 6.9 Ki 3
POSTYOWAJZBEMF 6.9 IC50 4
GQMKJIVMMQHGLX 6.9 Ki 2
GKRCHWBIEBSANV 6.9 Ki 3
VPNNTFDQKJOHAQ 6.9 Ki 2
APXAIXPMIFECKD 6.9 Ki 2
MFTQITSPGQORDA 6.9 IC50 9
CKYREKXNBZFCFF 6.9 Ki 2
AAOXQNKZMYOFJU 6.8 Ki 2
ALVYBVAQSFMTGH 6.8 Ki 3
FZYMAUQRNZROJG 6.8 Ki 3
MSOTYSLKONXWAT 6.8 Ki 3
QHGDTGBHXYZJHD 6.8 Ki 2
TYQUIMNJDNFTJV 6.8 Ki 2
WVTBQBGYKOVDJN 6.8 Ki 2
XMSAWCPABLSFFM 6.8 Ki 6
GHYMNVIBQBGLDY 6.8 Ki 2
LTXLJGIDFWWEQI 6.8 Ki 4
OUPJOWDHCXNNFZ 6.8 Ki 2
PCIBKAPYDVLZRH 6.8 Ki 3
MGOLGCRWUARCLB 6.8 Ki 2
SVDSEBLMCDOJKU 6.8 Ki 3
GVDWENUEEMSFBD 6.8 Ki 2
KIGJPKCRBSBFNE 6.8 Ki 2
VWKDMGIRFQHGHQ 6.8 Ki 3
BKMXGSZQEWHCJH 6.8 IC50 4
COPFNINVTDIILJ 6.8 Ki 3
GOERAAJVARXHDP 6.8 IC50 4
GUFLDWJZHZVTCO 6.8 Ki 2
WFUWFCPVIJPOGN 6.8 Ki 2
UTYMFQPKWLTXJA 6.7 Ki 3
CFSQPEBVGUSQII 6.7 Ki 5
DJPZZIPELMVWNS 6.7 Ki 5
QNQQOCOEVIOOFR 6.7 Ki 3
AACVRGGQVLDYDM 6.7 Ki 4
BNADKFGPICFCAD 6.7 Ki 2
DLXQMELVHFKJOP 6.7 Ki 3
JBHISGPWLXASFE 6.7 IC50 2
IPIVVFVBOCKVJN 6.7 Ki 3
WCFWDBPDMBXMTQ 6.7 Ki 3
2D structure