Target Details
UniProt ACP00749
Gene SymbolPLAU
Protein NameUrokinase-type plasminogen activator
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00051 (Kringle) PF00089 (Trypsin)
Summary
  • Multi-target molecules 256
  • Clinical molecules 4
  • Avg pChEMBL 6.99
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (256)
InChIKey pChEMBL Type Targets Clinical
MUPHEXMZSXMJJT 7.6 Ki 6
DARQQJKHXPXSRO 7.6 Ki 4
DARQQJKHXPXSRO 7.6 Ki 4
HUYQYLFFFNSAAX 7.6 Ki 3
VGQFBYXDHFTAHX 7.6 Ki 6
KORAEYDOYHOKIN 7.6 Ki 4
FWTQOPWAMQXIMI 7.6 Ki 3
BKTRHCGXWUYGAQ 7.5 Ki 2
DXFJLEXWZBCHSJ 7.5 Ki 3
XVWWDCXPGPSOQP 7.5 Ki 3
QEWPWXLSDLXYFF 7.5 Ki 3
MINVOLKUPZPDNX 7.5 Ki 3
GRQLDCHTDNYVQI 7.5 Ki 2
VHCWDBADFMDZND 7.5 Ki 2
FDCBFBSFHLWFFU 7.5 Ki 6
WUQXRUBSQOUYBJ 7.5 IC50 2
PSVQYWPWPKKKLA 7.5 IC50 6
YBSXFYTXULBNOE 7.5 Ki 6
YWZCPTFDCKPYIP 7.5 Ki 4
MIDRZAUOYQDRRT 7.4 Ki 2
DDKWYWKPXNAXSP 7.4 Ki 2
PTCHEYWURWFAME 7.4 Ki 5
BZRUPWYKAWYNCC 7.4 Ki 5
SJOGQFLRNCUNDK 7.4 Ki 5
FWEWLZSBDNPNAD 7.3 Ki 3
WQVBAYOMZJYFJK 7.3 IC50 8
FEPIUXBUJVISNN 7.3 Ki 2
MXIQAZDBFHHAPP 7.3 Ki 2
XRHANBWAKSYPEN 7.3 Ki 4
OOFRCFJPOZMMHV 7.3 Ki 3
VIZNZQTZRMTYPZ 7.3 Ki 4
IBHLYVDUKHZEBW 7.3 IC50 2
GWGDIYWVTCPPIK 7.3 IC50 2
HYEXCVYTGASYJN 7.3 IC50 2
QHOGUHKKMFDODA 7.3 Ki 6
DBQIGPPIAXXZLB 7.2 Ki 2
BHABIMFLZUWIMZ 7.2 Ki 2
NVXNLVNWFQMECM 7.2 IC50 2
QFJOOWSJASQPAX 7.2 IC50 7
RNMLDMHQKBIMRF 7.2 Ki 3
APXAIXPMIFECKD 7.2 Ki 2
BVTBOJXEAPSOEB 7.2 Ki 6
JECHDKUWRBFZLB 7.1 Ki 5
OPOYAWWWOKBVEB 7.1 Ki 6
OPOYAWWWOKBVEB 7.1 Ki 6
KLVFDMVKNCAXRG 7.1 Ki 2
NJJGNTZNFLYOMP 7.1 Ki 3
IEKKKOCYKOJJBP 7.0 Ki 3
PYBQUZRFYXFVJH 7.0 Ki 2
ONJMNFUCIIFBMG 7.0 Ki 2
2D structure