Target Details
UniProt ACP00749
Gene SymbolPLAU
Protein NameUrokinase-type plasminogen activator
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00051 (Kringle) PF00089 (Trypsin)
Summary
  • Multi-target molecules 256
  • Clinical molecules 4
  • Avg pChEMBL 6.99
Associated Diseases (1)
Top Co-occurrence Targets
Active Molecules (256)
InChIKey pChEMBL Type Targets Clinical
WLDWWFXJFODOTC 9.3 Ki 7
CSWQJKHBMACTGB 9.2 Ki 6
SXVLRRZGNNRRFR 9.1 IC50 2
KAUYBZJFBAONCO 9.1 Ki 6
ONSBFNASIDWXPA 8.7 Ki 5
FIKPJJWWHHKTHI 8.7 Ki 2
ITFFOKFQKAACGD 8.6 Ki 2
LLKJHSDOKTVQNQ 8.5 IC50 2
KXIPWEMRKHDRAH 8.5 IC50 2
XELNXCJTRAIQOD 8.5 Ki 4
BXSDRFZOPSIGSI 8.4 IC50 4
VCVSFHZQGWZRGK 8.4 IC50 4
DZZJIIDXFNEDSI 8.4 IC50 3
WHOCSXXAQICVLG 8.4 IC50 3
CZRSUKWCMUIVJO 8.3 Ki 3
JYLDIRMFPPDHNN 8.3 IC50 2
FMQAKCLMDYHTJC 8.2 IC50 2
VXFFMDVLGNSKLD 8.2 IC50 2
ORVXTXWYNQMIKW 8.2 IC50 2
QDCFZMDANJYLAS 8.2 IC50 2
LVNMYQLXKMSQTG 8.2 Ki 3
LVNMYQLXKMSQTG 8.2 Ki 3
IBGRQIRGZCRMEE 8.2 IC50 2
SCFDAWOKUNONKP 8.2 IC50 2
CTDHLROQTKJDLK 8.2 IC50 4
QJNHUFOFEMCMGR 8.1 Ki 4
CSTAEACZUNFQMP 8.1 IC50 3
GAVRMVQHHVMXFD 8.1 Ki 11
ZLSGXUVBYIIXKU 8.1 Ki 5
HLWKBMWAJJZWIT 8.1 Ki 5
FEKRWNWZMOSVBX 8.1 Ki 6
HNGQAWXKSWVXIP 8.0 Ki 2
RTPDDFLFZXREMW 8.0 Ki 3
GIXXCPBLBWRNFX 8.0 IC50 2
RFUDJRCNYAUEMT 7.9 IC50 2
BCXSNIMTARZGHJ 7.9 Ki 4
FEKRWNWZMOSVBX 7.9 Ki 3
GOBXSXIHPUGHDS 7.8 Ki 6
NTNRVRBIIZBTBR 7.8 IC50 8
RCWPAPFNFNQLML 7.8 Ki 3
CMCDWLMEDRBWIR 7.7 Ki 2
VGKVWATXDPBYQQ 7.7 Ki 5
JKZBIUMNKJTCCD 7.7 IC50 2
HECONMODEBIAKY 7.7 IC50 9
MMMVHDBARFPCLX 7.7 Ki 6
NKADRYHVDUCFQU 7.7 Ki 4
NKADRYHVDUCFQU 7.7 Ki 4
RHEKWNPDSIWZKZ 7.7 IC50 8
ZNOKJHWJKULOGM 7.7 IC50 2
GKFHRQMCFNIZHA 7.7 Ki 4
2D structure