Target Details
| UniProt AC | P00748 |
|---|---|
| Gene Symbol | F12 |
| Protein Name | Coagulation factor XII |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00008 (EGF) PF00039 (fn1) PF00040 (fn2) PF00051 (Kringle) PF00089 (Trypsin) |
Summary
- Multi-target molecules 175
- Clinical molecules 0
- Avg pChEMBL 6.64
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (175)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UXTLTIOXBOHGKL
|
6.2 | IC50 | 3 | — | |
WDKFWBZIMKMRIR
|
6.2 | IC50 | 2 | — | |
WZFGKOMTANPZBQ
|
6.2 | IC50 | 2 | — | |
XEJIXVCRPCLTGX
|
6.2 | IC50 | 3 | — | |
XQRKYMOJJOXHBZ
|
6.2 | IC50 | 2 | — | |
XZQLWSAQKCFLPX
|
6.2 | IC50 | 2 | — | |
YCUHYXGBQOXOJG
|
6.2 | IC50 | 6 | — | |
YSHBWHHQCNCYQM
|
6.2 | IC50 | 2 | — | |
ZKYUOZOXYNXLAA
|
6.2 | IC50 | 4 | — | |
DTIUMOLBWQXRPH
|
6.2 | Ki | 3 | — | |
YLUMVCNEFHTQHD
|
6.2 | IC50 | 3 | — | |
OBYVXAUONRVYHA
|
6.1 | Ki | 2 | — | |
GCEWJBIDLIIRAB
|
6.1 | IC50 | 2 | — | |
IWNWXPRWSFWNMU
|
6.1 | Ki | 5 | — | |
UJHCYBGLPMMJDH
|
6.1 | IC50 | 3 | — | |
BIEYFOHSWAIQDF
|
6.1 | IC50 | 5 | — | |
GWZGMZVWURNLOZ
|
6.1 | Ki | 4 | — | |
IHUNZLYUFXYPJH
|
6.1 | IC50 | 2 | — | |
BVZHCUOVJATBQP
|
6.1 | Ki | 5 | — | |
SIISFRLGYDVIRG
|
6.1 | Ki | 2 | — | |
GTLWZDWHNMMHMP
|
6.0 | IC50 | 2 | — | |
CSZFJKLNCKEZQL
|
6.0 | IC50 | 3 | — | |
UWCPWBIMRYXUOU
|
6.0 | Ki | 3 | — | |
YFOBXIFGQIGNEC
|
6.0 | IC50 | 2 | — | |
XKJPYUYSROHYIL
|
6.0 | IC50 | 2 | — |