Target Details
| UniProt AC | P00748 |
|---|---|
| Gene Symbol | F12 |
| Protein Name | Coagulation factor XII |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00008 (EGF) PF00039 (fn1) PF00040 (fn2) PF00051 (Kringle) PF00089 (Trypsin) |
Summary
- Multi-target molecules 175
- Clinical molecules 0
- Avg pChEMBL 6.64
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (175)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RVSYWOORIBXTII
|
6.6 | IC50 | 2 | — | |
RUGKDKWVOXRCGI
|
6.5 | Ki | 2 | — | |
NHXDITCQCUWVEW
|
6.5 | IC50 | 2 | — | |
JPJWLXDMTIOTSV
|
6.5 | IC50 | 2 | — | |
QKNUHBOQEJLPLK
|
6.5 | IC50 | 2 | — | |
SESLACGWCLIGCW
|
6.5 | Ki | 2 | — | |
UHZMCBKFZIOFLI
|
6.5 | IC50 | 8 | — | |
GKBXJOCPZBRUIG
|
6.4 | IC50 | 4 | — | |
ITJOJULATKBZRP
|
6.4 | IC50 | 2 | — | |
BJSIWIFJSRFHPS
|
6.4 | Ki | 6 | — | |
ZCDZQESCUOZOOO
|
6.4 | IC50 | 8 | — | |
GLLWHIMOHBWLKF
|
6.3 | IC50 | 2 | — | |
ZAFULIRXGRRKIP
|
6.3 | IC50 | 3 | — | |
GHJUQPDHYJIXSP
|
6.3 | IC50 | 2 | — | |
XATHBXYKVIAZOR
|
6.3 | Ki | 3 | — | |
ZNIQLYYOYYLSEW
|
6.3 | IC50 | 3 | — | |
OGCGKERBEQPTBU
|
6.3 | Ki | 3 | — | |
CGCVHJCZBIYRQC
|
6.2 | Ki | 2 | — | |
QCJKXYYLKAMQSD
|
6.2 | Ki | 5 | — | |
BAPGDFQYYPBNAG
|
6.2 | IC50 | 2 | — | |
BGYKTPXLTQILOF
|
6.2 | IC50 | 2 | — | |
BKGCNONNVNNPCJ
|
6.2 | IC50 | 2 | — | |
CSOIEWKCRIAOFP
|
6.2 | IC50 | 2 | — | |
CUJAMZMFVUMLMN
|
6.2 | IC50 | 3 | — | |
DVKBAFOJFMJCAO
|
6.2 | IC50 | 2 | — | |
FUQWXNUBICSJBF
|
6.2 | IC50 | 4 | — | |
GANUYKJXFODNNH
|
6.2 | IC50 | 2 | — | |
GXJGGSLRORREAO
|
6.2 | IC50 | 2 | — | |
HDPSRBDROYEPJE
|
6.2 | IC50 | 3 | — | |
HMMQIOFQLZWHKO
|
6.2 | IC50 | 2 | — | |
IGCDDPNPYAFVCA
|
6.2 | IC50 | 2 | — | |
IVQXOYFHEXATGH
|
6.2 | IC50 | 3 | — | |
JBHALIPUGWBOFZ
|
6.2 | IC50 | 2 | — | |
KGSRYOUTAFUTIJ
|
6.2 | IC50 | 3 | — | |
KPFQKUFJYSBYBL
|
6.2 | IC50 | 3 | — | |
LWFLIRIWEPBXFX
|
6.2 | Ki | 4 | — | |
MBFJFSDXDXLAQN
|
6.2 | IC50 | 2 | — | |
NUXYYWOWNFEMNH
|
6.2 | Ki | 2 | — | |
PIUDHEFNICCZME
|
6.2 | IC50 | 2 | — | |
QCLWJMUFTKLIAE
|
6.2 | IC50 | 2 | — | |
QEKIKQCZDOHATQ
|
6.2 | IC50 | 2 | — | |
QSWJYWCLHVAJEZ
|
6.2 | IC50 | 2 | — | |
RJGXWYMMSWXDBY
|
6.2 | IC50 | 4 | — | |
RRDABEWIPOYJNA
|
6.2 | IC50 | 2 | — | |
RVIHDYFOYNJDSF
|
6.2 | IC50 | 2 | — | |
RWQRQTTUCTXRQC
|
6.2 | IC50 | 4 | — | |
SJKSASQLXWHGFH
|
6.2 | IC50 | 4 | — | |
SOTJCXRFTOZWTE
|
6.2 | IC50 | 2 | — | |
SWVWAZLEARISBG
|
6.2 | IC50 | 2 | — | |
UPPRVHQOSXWZLP
|
6.2 | IC50 | 3 | — |