Target Details
| UniProt AC | P00748 |
|---|---|
| Gene Symbol | F12 |
| Protein Name | Coagulation factor XII |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00008 (EGF) PF00039 (fn1) PF00040 (fn2) PF00051 (Kringle) PF00089 (Trypsin) |
Summary
- Multi-target molecules 175
- Clinical molecules 0
- Avg pChEMBL 6.64
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (175)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KSAWJQXHHNRNMK
|
6.7 | IC50 | 2 | — | |
UKMUINAUAULENG
|
6.7 | Ki | 2 | — | |
CCUGLTODPQTEBR
|
6.7 | IC50 | 7 | — | |
WUANWHWUHPZKMS
|
6.7 | IC50 | 2 | — | |
AIRGERSZASMAFK
|
6.7 | IC50 | 2 | — | |
AYQRIBJCWHYQNN
|
6.7 | IC50 | 2 | — | |
CKNZDXKTBCVSIY
|
6.7 | IC50 | 2 | — | |
CQDVUJSXYFSSHR
|
6.7 | IC50 | 4 | — | |
CSNSELBEUILYAV
|
6.7 | IC50 | 2 | — | |
CYDSMQBZTXOTJO
|
6.7 | IC50 | 2 | — | |
DLIVTYIYTMUJNA
|
6.7 | IC50 | 4 | — | |
IFOVGASEQCOJAP
|
6.7 | IC50 | 2 | — | |
IPMBKJBCZMJJID
|
6.7 | IC50 | 2 | — | |
JRGKULXTRBRGAB
|
6.7 | IC50 | 2 | — | |
KITXJRBAWLMDQM
|
6.7 | IC50 | 3 | — | |
LAEZPLWSRMVDKT
|
6.7 | IC50 | 5 | — | |
LEOZSBNDFVBQQT
|
6.7 | IC50 | 5 | — | |
LRIAAYQSNNESBQ
|
6.7 | IC50 | 2 | — | |
MABZHGPFQUEHHT
|
6.7 | IC50 | 4 | — | |
MAMDUCKALBRXSZ
|
6.7 | IC50 | 2 | — | |
NDQYBUYVXIWGNJ
|
6.7 | IC50 | 2 | — | |
OGEBHANRXXUPQA
|
6.7 | IC50 | 3 | — | |
OJOAPDZWILJFFF
|
6.7 | IC50 | 2 | — | |
PGGPSANDIMXVMM
|
6.7 | IC50 | 2 | — | |
PHLLDHUJAMWXHD
|
6.7 | IC50 | 3 | — | |
PIUDHEFNICCZME
|
6.7 | IC50 | 2 | — | |
PRHIFYJJLKNAIF
|
6.7 | IC50 | 2 | — | |
PUSHOPRQHUASRC
|
6.7 | IC50 | 2 | — | |
QDOYQXPRWRGBKF
|
6.7 | IC50 | 3 | — | |
QXBVZJVFQPOKBL
|
6.7 | IC50 | 2 | — | |
RBVSANJGHRPNCU
|
6.7 | IC50 | 2 | — | |
RETOSFBTHJWCPW
|
6.7 | IC50 | 3 | — | |
RJQLFWVERDFMFU
|
6.7 | IC50 | 4 | — | |
RMNYKKOMVGKWMF
|
6.7 | IC50 | 3 | — | |
RTTUBFUCOXOZCQ
|
6.7 | IC50 | 4 | — | |
SBFVHGJSVOMQJH
|
6.7 | IC50 | 4 | — | |
SXIFTOXSOJHIGC
|
6.7 | IC50 | 3 | — | |
SXVRJEWRROULBO
|
6.7 | IC50 | 4 | — | |
UMCJVSRVNNGRDY
|
6.7 | IC50 | 4 | — | |
UMCJVSRVNNGRDY
|
6.7 | IC50 | 6 | — | |
UMFFCYDWHBQNPV
|
6.7 | IC50 | 4 | — | |
UXQJFMQHQIXERQ
|
6.7 | IC50 | 2 | — | |
WHPTVTWMXGFSRJ
|
6.7 | Ki | 2 | — | |
XEVLXXSTUOLYHZ
|
6.7 | IC50 | 2 | — | |
YGRNPRKEECJLCM
|
6.7 | IC50 | 3 | — | |
YHMGDTWUZGOVRL
|
6.7 | IC50 | 2 | — | |
ZGZPKQSHBQJIGW
|
6.7 | IC50 | 2 | — | |
WLZYFEBXZVJFMV
|
6.7 | IC50 | 2 | — | |
KWPACVJPAFGBEQ
|
6.6 | Ki | 2 | — | |
HUOMJWOJQZRJRS
|
6.6 | IC50 | 8 | — |