Target Details
| UniProt AC | P00748 |
|---|---|
| Gene Symbol | F12 |
| Protein Name | Coagulation factor XII |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00008 (EGF) PF00039 (fn1) PF00040 (fn2) PF00051 (Kringle) PF00089 (Trypsin) |
Summary
- Multi-target molecules 175
- Clinical molecules 0
- Avg pChEMBL 6.64
KEGG Pathways (1)
Associated Diseases (2)
Active Molecules (175)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GQEQKTGRIPEAKW
|
8.1 | Ki | 2 | — | |
OGTUYARYUMRJAT
|
8.0 | Ki | 2 | — | |
JLUGWHXZCKLPBY
|
8.0 | Ki | 2 | — | |
QMRJOIUGPCVZPH
|
7.7 | Ki | 6 | — | |
VQSLCEFIEDDAEK
|
7.6 | IC50 | 2 | — | |
JSYAAQWLHIRCII
|
7.5 | IC50 | 2 | — | |
CYAQTWKBNHAHHY
|
7.5 | IC50 | 2 | — | |
VEBLIIOSJXGVAW
|
7.5 | Ki | 3 | — | |
BZGZTAKGLPGMAV
|
7.3 | IC50 | 3 | — | |
VCSUDCIPCNCOHV
|
7.3 | IC50 | 3 | — | |
ADOGWSXMKPYQAU
|
7.3 | IC50 | 4 | — | |
BKGCNONNVNNPCJ
|
7.3 | IC50 | 2 | — | |
COGDLYORVLPAJK
|
7.3 | IC50 | 3 | — | |
CYDSMQBZTXOTJO
|
7.3 | IC50 | 2 | — | |
FANJUXPUAIHWDE
|
7.3 | IC50 | 5 | — | |
FCXNRNCBQJLWDJ
|
7.3 | IC50 | 3 | — | |
HSNORKMSWCSMOD
|
7.3 | IC50 | 2 | — | |
JRXMHNDYGQNYAI
|
7.3 | IC50 | 4 | — | |
KHKMNGWOVOQDJO
|
7.3 | IC50 | 2 | — | |
MWDLRAJKBFJGKK
|
7.3 | IC50 | 2 | — | |
NDQYBUYVXIWGNJ
|
7.3 | IC50 | 2 | — | |
NDQYBUYVXIWGNJ
|
7.3 | IC50 | 3 | — | |
PGGPSANDIMXVMM
|
7.3 | IC50 | 3 | — | |
VFEVHMYHGBXCLM
|
7.3 | IC50 | 3 | — | |
VQSLCEFIEDDAEK
|
7.3 | IC50 | 2 | — | |
VZCLQKXKPFPMJM
|
7.3 | IC50 | 3 | — | |
WPHHTTMLRJZZSE
|
7.3 | IC50 | 5 | — | |
XGBLRGJOWPDUDW
|
7.3 | IC50 | 3 | — | |
YXPALMWXBGWOBZ
|
7.3 | IC50 | 3 | — | |
SYHAFKBWNBYQST
|
7.2 | Ki | 3 | — | |
KGRJPLRFGLMQMV
|
7.2 | Ki | 2 | — | |
LFZPKEYIGZKMGC
|
7.1 | IC50 | 2 | — | |
UHIWVKZCJPLNNG
|
7.0 | IC50 | 2 | — | |
DZGOQOXWBUEYTK
|
7.0 | IC50 | 2 | — | |
AHBGDSREPWVVFA
|
7.0 | IC50 | 2 | — | |
LGYDKGKNEZTQLV
|
7.0 | IC50 | 2 | — | |
MRKFVLTUFONGMP
|
7.0 | Ki | 2 | — | |
MQQNFDZXWVTQEH
|
7.0 | Ki | 11 | — | |
QQRQFIXRVWJLNT
|
7.0 | Ki | 10 | — | |
RNYFAJPMYTZRIV
|
7.0 | IC50 | 4 | — | |
BAQBCWWGOQNMJV
|
7.0 | IC50 | 2 | — | |
OOSAWCAECZEMCW
|
7.0 | Ki | 6 | — | |
LDGAAMMSVIUSAT
|
6.9 | IC50 | 2 | — | |
CAVJGRPSJPRJNJ
|
6.9 | IC50 | 2 | — | |
LOMJHEAYYYPWDO
|
6.9 | IC50 | 2 | — | |
AKDDPMDJFJJCDW
|
6.8 | IC50 | 16 | — | |
FLJAMCIHLYTQCT
|
6.8 | IC50 | 4 | — | |
WINMHXQNIIDEPT
|
6.8 | IC50 | 2 | — | |
ZAQVKSRGAWOLLX
|
6.8 | Ki | 2 | — | |
HCCRRLVJBLDSLL
|
6.8 | IC50 | 2 | — |