Target Details
| UniProt AC | P00734 |
|---|---|
| Gene Symbol | F2 |
| Protein Name | Prothrombin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00594 (Gla) PF00051 (Kringle) PF09396 (Thrombin_light) PF00089 (Trypsin) |
Summary
- Multi-target molecules 1,259
- Clinical molecules 4
- Avg pChEMBL 7.37
KEGG Pathways (8)
Associated Diseases (2)
Active Molecules (1,259)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RMYIJADBJGXIMY
|
7.8 | Ki | 2 | — | |
DPEVDPDGUAGUHE
|
7.8 | IC50 | 4 | — | |
JSZQNSABSYYEPQ
|
7.8 | IC50 | 2 | — | |
QLPNTZLPNDVFJT
|
7.8 | Ki | 2 | — | |
UWMOBFHBRYCOPF
|
7.8 | IC50 | 3 | — | |
VDEXCODLWRXIIG
|
7.8 | IC50 | 4 | — | |
VKYVGNOZMWMZDF
|
7.8 | IC50 | 2 | — | |
XYHQRSYCQQCWPT
|
7.8 | IC50 | 3 | — | |
ZVZKYABQRFIIAV
|
7.8 | IC50 | 3 | — | |
QAIZMIBCSNGQKN
|
7.8 | IC50 | 5 | — | |
RXCJPCHXBRDPDW
|
7.8 | Ki | 2 | — | |
IAUZEBLXCOCAFL
|
7.8 | Ki | 2 | — | |
VOALXMVXTCHJGT
|
7.8 | IC50 | 2 | — | |
YIMMYYIRSBUOIA
|
7.8 | Ki | 4 | — | |
JCHJGPGQBMUBTD
|
7.8 | Ki | 2 | — | |
DKFBIZDHPKUBIT
|
7.8 | IC50 | 5 | — | |
GOZOOJYBIIQGLI
|
7.8 | IC50 | 3 | — | |
KAGLWQUWUNBAOO
|
7.8 | IC50 | 5 | — | |
KXTBCHXZWNKXAC
|
7.8 | Ki | 2 | — | |
RPWMNCDNXZFZIK
|
7.8 | IC50 | 4 | — | |
GYZAJGLGNWNLGL
|
7.7 | IC50 | 2 | — | |
HGZAKQZABFGBLF
|
7.7 | IC50 | 2 | — | |
HGZDLWBCOWFXST
|
7.7 | IC50 | 3 | — | |
JENOLOFVMYLCBZ
|
7.7 | IC50 | 3 | — | |
TVKPLGVIMIGLSZ
|
7.7 | Ki | 4 | — | |
TYJWNUCOFLGCGZ
|
7.7 | IC50 | 4 | — | |
XHOLNRLADUSQLD
|
7.7 | IC50 | 2 | — | |
YSHIHBNJUPKMRT
|
7.7 | IC50 | 4 | — | |
BDYQCMIJBWOCAH
|
7.7 | IC50 | 2 | — | |
FRPFDONKAHIRLY
|
7.7 | IC50 | 2 | — | |
HJPWRDMWCBCSDO
|
7.7 | Ki | 5 | — | |
KXTBCHXZWNKXAC
|
7.7 | Ki | 2 | — | |
PREVZZBJVCTDTQ
|
7.7 | IC50 | 5 | — | |
XJDVJJDJQXRAOB
|
7.7 | Ki | 4 | — | |
BDLMBQRBNPDCSS
|
7.7 | IC50 | 2 | — | |
CWEMMPPJSUYKOM
|
7.7 | IC50 | 2 | — | |
HGNSKHRWYAJRBQ
|
7.7 | Ki | 5 | — | |
ILRJJEMRKWAJMZ
|
7.7 | IC50 | 2 | — | |
QHRDZTQSQGOQEL
|
7.7 | IC50 | 2 | — | |
XTUJNPODMRCIHC
|
7.7 | IC50 | 4 | — | |
FRPFDONKAHIRLY
|
7.7 | IC50 | 2 | — | |
HLLDKSBRPSVLQJ
|
7.7 | IC50 | 2 | — | |
MTPIBEHXUUEJRW
|
7.7 | Ki | 2 | — | |
VKNTYOZSHHKHTK
|
7.7 | Ki | 3 | — | |
WXVYOXMMXUJYLQ
|
7.7 | IC50 | 4 | — | |
FXRJBDKVWJJJSK
|
7.6 | Ki | 2 | — | |
GEOOUXGQTSKLIU
|
7.6 | IC50 | 2 | — | |
OLFJSYFEVMJTBF
|
7.6 | IC50 | 2 | — | |
OQYJSEGEYSKAGD
|
7.6 | IC50 | 2 | — | |
PLAJAOHXCUUQEL
|
7.6 | IC50 | 3 | — |