Target Details
UniProt ACP00734
Gene SymbolF2
Protein NameProthrombin
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00594 (Gla) PF00051 (Kringle) PF09396 (Thrombin_light) PF00089 (Trypsin)
Summary
  • Multi-target molecules 1,259
  • Clinical molecules 4
  • Avg pChEMBL 7.37
Top Co-occurrence Targets
Active Molecules (1,259)
InChIKey pChEMBL Type Targets Clinical
FHVWKHLVLPLXNR 8.1 Ki 2
JDXUSWQJCGTBLN 8.1 IC50 2
LMZXSQIAAPRXML 8.1 Ki 2
BNQKKJULGXDFIQ 8.0 Ki 2
UPFBONOEYAFXQG 8.0 Ki 5
FCTCJAGJUHHZDO 8.0 IC50 3
QGNIEHVRQPFGKU 8.0 Ki 2
RBROQTNENUBMPK 8.0 Ki 2
ODAGEWXXQNKGPN 8.0 Ki 3
QWTIOQGNSLCKBH 8.0 IC50 3
GMTPFEPAXXLLCG 8.0 Ki 4
IFEIYEIENSCXHQ 8.0 IC50 2
JENOLOFVMYLCBZ 8.0 IC50 4
LHVRINJTNXVOIY 8.0 IC50 2
QINGREKOIHZHSD 8.0 IC50 2
QYHLFIWGLVWPSH 8.0 IC50 2
PVTLJXXAPWJMAT 8.0 IC50 2
GYNIHHFDCVUJCX 8.0 Ki 4
QOLVMRURXPRFJX 8.0 Ki 2
XJJMRYCODRNFRY 8.0 Ki 5
GVACGRWTTRFLEX 7.9 IC50 4
BCXSNIMTARZGHJ 7.9 Ki 4
PALUIMPWPYLQAY 7.9 Ki 4
PBMZSYYXSHEKKY 7.9 IC50 4
RNMRZBAGAMQNNF 7.9 Ki 2
XKFOQXQRMWVYJC 7.9 IC50 2
ZJJGXYMWSZBKRL 7.9 IC50 2
OLFYUUPVCGARIA 7.9 IC50 4
UGKVIJMVQRJDEZ 7.9 Ki 2
IJPKHEGDEHMVNS 7.9 Ki 3
MIMFPYZFIMECLR 7.9 IC50 2
WBPLJGAAZCZXSP 7.9 IC50 5
YJNVYIQRUCUHIU 7.9 IC50 2
BPQSFHAKWPDIHD 7.9 Ki 4
NZEAENHOWXTKPM 7.9 IC50 5
VMWSTSFZJLCRPU 7.9 Ki 4
CZYFQAJCCZGMEU 7.8 IC50 3
NGRWSGCZGGUEEZ 7.8 IC50 3
UAKRLLAUOQEYFN 7.8 IC50 3
CDRQZRZODAGYKU 7.8 Ki 4
BQDYQUZLQVWWMF 7.8 IC50 4
JVXBUVJQTIKERQ 7.8 IC50 5
CDPROXZBMHOBTQ 7.8 Ki 4
CDPROXZBMHOBTQ 7.8 Ki 2
DCIWCRNLCDDMQZ 7.8 Ki 2
FXSYQODCNXHQNQ 7.8 IC50 4
HZXNJMYMOIYCPJ 7.8 IC50 2
MLVRJRSVNIXHHG 7.8 IC50 2
OCNKSJHQWUSIRB 7.8 IC50 5
OFNBWUOTBUVGEV 7.8 IC50 2
2D structure