Target Details
UniProt ACP00734
Gene SymbolF2
Protein NameProthrombin
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00594 (Gla) PF00051 (Kringle) PF09396 (Thrombin_light) PF00089 (Trypsin)
Summary
  • Multi-target molecules 1,259
  • Clinical molecules 4
  • Avg pChEMBL 7.37
Top Co-occurrence Targets
Active Molecules (1,259)
InChIKey pChEMBL Type Targets Clinical
VFEVHMYHGBXCLM 8.5 IC50 3
WJAIHAMGHSKLNB 8.5 IC50 2
WMVZLWYOHAUGMC 8.5 IC50 3
WPHHTTMLRJZZSE 8.5 IC50 5
WYPYYUPYCYVRGI 8.5 IC50 2
XCVKPLFBAXRCKB 8.5 IC50 2
XEJIXVCRPCLTGX 8.5 IC50 3
YGRNPRKEECJLCM 8.5 IC50 3
YNXJBBUWTCLOKJ 8.5 Ki 2
YUGVXCKQXRQZMT 8.5 IC50 4
ZKYUOZOXYNXLAA 8.5 IC50 4
DKOQLRVNWZHTGN 8.5 Ki 2
RYQMPGLCCOYWRL 8.5 Ki 3
WEZCXOSTNFUHCF 8.5 IC50 3
ZPSJUJRQJVQURK 8.5 Ki 2
FQFUSWODGXTQQH 8.5 Ki 5
CTJBFJRLIYRRCN 8.5 Ki 3
KIOBRCOIPVZTCH 8.5 Ki 2
NYKOPIYZICLSFY 8.5 Ki 2
AABZTMRZWJMBNH 8.4 IC50 2
FVYGXQLKUXZGOL 8.4 Ki 2
BUIUXNUKSBOYIU 8.4 Ki 2
UERHFNVGKAURME 8.4 Ki 2
DXCOONBXASCQJO 8.4 IC50 4
GHCPCZIUEYRYJT 8.4 Ki 2
GMKHQRCPNMGCIX 8.4 IC50 2
OUFALBVXADUJCB 8.4 IC50 2
TVZGEZJAWHKQJW 8.4 Ki 2
WXLILDXQUZIWFM 8.4 Ki 2
JXHWVKOKYDAROD 8.4 Ki 4
USJGYEQJWLDDDM 8.4 IC50 7
WLDWWFXJFODOTC 8.4 Ki 7
JCTRHKZXDDIGIB 8.4 Ki 2
FNTZDDYIJOPMAJ 8.4 Ki 2
UHRIYOJEACOYON 8.4 IC50 3
HSCBDDXIIWYLQX 8.3 Ki 2
YBSJFWOBGCMAKL 8.3 IC50 5
GFXFOCFFDUYUAQ 8.3 Ki 5
VYJOAYZRCNHDNG 8.3 Ki 6
RROGCGMHOWNSLD 8.3 IC50 2
ANSWPKCJQAZJTJ 8.3 Ki 3
OAQVACIWUZCUCP 8.3 Ki 2
UHSOJTIMDDIBQO 8.3 IC50 5
YNGAKUMMINESNS 8.3 Ki 2
YWKFVICYLBEIJR 8.3 Ki 2
CEAMGXQGUYMUIE 8.3 Ki 2
CPBDFCXKCBYWQN 8.3 IC50 5
DFDTTXLYOCLPSE 8.3 Ki 2
LAGUWJUZJRIYRI 8.3 IC50 2
NSRPFWUFZRMLQX 8.3 IC50 2
2D structure