Target Details
UniProt ACP00734
Gene SymbolF2
Protein NameProthrombin
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00594 (Gla) PF00051 (Kringle) PF09396 (Thrombin_light) PF00089 (Trypsin)
Summary
  • Multi-target molecules 1,259
  • Clinical molecules 4
  • Avg pChEMBL 7.37
Top Co-occurrence Targets
Active Molecules (1,259)
InChIKey pChEMBL Type Targets Clinical
DSEQCUGXKCOSSU 8.9 IC50 5
OVQWFZKRHDTPOD 8.9 IC50 7
NZEDSGTYZINZBH 8.8 Ki 3
OAZBEQQNMLSDQD 8.8 IC50 2
MJWDBCUSOIFRIS 8.8 IC50 2
BRZYOTMFHLERHD 8.8 IC50 17 Yes
KWPACVJPAFGBEQ 8.8 IC50 2
SEULIANDYJKOAE 8.8 Ki 2
VZFTWWJAUZOJDH 8.8 Ki 2
WJPYSLNVRNBWAJ 8.8 Ki 2
WJPYSLNVRNBWAJ 8.8 Ki 2
AUHROPMDFWDFRD 8.8 IC50 2
KLBBHAHSBBTWTB 8.8 Ki 3
MBPIOWHYJVTSDB 8.8 Ki 3
OGIUPCNSPIXREF 8.8 Ki 2
CETVCAHONSWCPC 8.8 Ki 2
HQFKZMCNWILBNJ 8.8 IC50 3
KBJGRHGRZYRRHG 8.8 Ki 6
NEEBGCAKJPDPFV 8.8 Ki 5
PKBJUALJQNSPHR 8.8 Ki 2
RIUCWNRPWWTWOU 8.8 Ki 3
VZFNTNJRDFGPHL 8.8 Ki 4
GJKMIUMNDMWVGF 8.8 IC50 5
HCHRFTFHZHSKTG 8.7 Ki 2
MTGQBIHLRYXSAD 8.7 IC50 3
XXDNJRMCHPIHOV 8.7 Ki 2
GFCCZFCZIXBOIU 8.7 IC50 2
MVBZVIDGYJOWNV 8.7 IC50 2
SMSISCIMPYBOQW 8.7 IC50 2
BKKXFHYCELTMFP 8.7 IC50 2
BOCSUPFQLFIHFX 8.7 IC50 4
CPRRWWFKLKISFM 8.7 Ki 4
FANJUXPUAIHWDE 8.7 IC50 5
FUBQFHITWDEUOJ 8.7 Ki 2
JRXMHNDYGQNYAI 8.7 IC50 4
KOQWYAURZBRJBF 8.7 IC50 2
LEOZSBNDFVBQQT 8.7 IC50 5
LPENKDDSJSQSIP 8.7 IC50 3
LPSWZZASPZFANL 8.7 IC50 2
PUHFAUFRLDIBFL 8.7 IC50 2
YMJHMJLNQLVUAV 8.7 Ki 2
ZLJLYLMJZPDBSJ 8.7 Ki 2
BIHPYGVYKSQDLA 8.7 IC50 5
FTIYOMFLKBWGLH 8.7 Ki 2
IMLVEYAVSNLRRR 8.7 IC50 2
KEEBLYWBELVGPQ 8.7 IC50 3
LJRHHCQQRGXIOI 8.7 Ki 2
MJWDBCUSOIFRIS 8.7 IC50 2
SKYLWGMFRJDRGN 8.7 Ki 2
OLKUSWOEHSSOHD 8.7 IC50 2
2D structure