Target Details
UniProt ACP00734
Gene SymbolF2
Protein NameProthrombin
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00594 (Gla) PF00051 (Kringle) PF09396 (Thrombin_light) PF00089 (Trypsin)
Summary
  • Multi-target molecules 1,259
  • Clinical molecules 4
  • Avg pChEMBL 7.37
Top Co-occurrence Targets
Active Molecules (1,259)
InChIKey pChEMBL Type Targets Clinical
JXHRRVFVLWWLCI 9.2 IC50 3
PIIUKKBKYNGKMK 9.2 IC50 3
PTYYNQHOHSWREY 9.2 IC50 2
ZASUNCQYGAHWBN 9.1 IC50 3
OELZFXTXLBIKDS 9.1 Ki 2
YELLYQPFWRBWSX 9.1 Ki 2
AQOWADPLFQHPQP 9.1 Ki 2
KBNWFXRFMYBDPZ 9.1 IC50 5
MJPRZTFMWHJGMK 9.1 Ki 6 Yes
DQTHQWDHVZBQHX 9.1 Ki 2
IGRCAZNQYXPQOS 9.1 Ki 2
WQFBTFLBEOJMDB 9.1 Ki 2
KAUYBZJFBAONCO 9.0 Ki 6
WRDBDBHZQFTGKU 9.0 Ki 2
AEAKGPDMUCEEJW 9.0 Ki 2
NUUVIYWKLAQTDU 9.0 IC50 2
BJIQNZYXWYUXEW 9.0 IC50 2
GTVCIMQDPDVJKE 9.0 Ki 2
YXSHAUMNJBEKLS 9.0 Ki 5
YXSHAUMNJBEKLS 9.0 Ki 3
BUGKCANFLDYYKD 9.0 IC50 6
CJPQDOALKKFQAR 9.0 IC50 2
FLJAMCIHLYTQCT 9.0 IC50 4
HKBDZTCNUODKEC 9.0 IC50 3
IELDEMOVCFANHT 9.0 IC50 5
KKJYVDXDZURHMA 9.0 Ki 5
LCMZZAYNITZFAI 9.0 Ki 4
MBNKUMIZUGCXRO 9.0 Ki 4
UVDLZNNZPDZTET 9.0 IC50 3
FBHFAKDPYSBTTM 9.0 IC50 3
JCYOSRSLFRMEPO 9.0 IC50 4
JOISFXBHQMBJET 9.0 Ki 2
LCCSPLBHNLGJIP 9.0 Ki 2
NTCIXIFCFSINOS 9.0 Ki 2
NXHSVNNVHFYXIB 9.0 Ki 2
VOIBTJMVYPMEOK 9.0 Ki 2
YLPFNSPUPARBLY 9.0 IC50 4
YTDWOXUEZRXCIH 9.0 Ki 2
OGPZZSRTWGPAJE 8.9 IC50 3
AWDJYEYUDBHRRD 8.9 Ki 5
ICMSWQUELAGTTR 8.9 IC50 2
IXWHJTMAJYJQMO 8.9 Ki 2
JSPAUBUYPPZXSG 8.9 IC50 17 Yes
LTVJYZXRRBSKBE 8.9 Ki 2
RACJERJJTUONSE 8.9 IC50 2
BTZOUFLORPKMGE 8.9 Ki 2
CROZVKXDALXCPS 8.9 IC50 6
GEGPKJUQKQSQAE 8.9 Ki 2
IDCKXHIGLKQWMM 8.9 Ki 4
VCWGHXLLKIVRCN 8.9 Ki 2
2D structure