Target Details
UniProt ACP00734
Gene SymbolF2
Protein NameProthrombin
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00594 (Gla) PF00051 (Kringle) PF09396 (Thrombin_light) PF00089 (Trypsin)
Summary
  • Multi-target molecules 1,259
  • Clinical molecules 4
  • Avg pChEMBL 7.37
Top Co-occurrence Targets
Active Molecules (1,259)
InChIKey pChEMBL Type Targets Clinical
KYTPBHITFYEVPE 7.0 Ki 2
OTGQDAVVEHBHSE 7.0 Ki 2
SYHAFKBWNBYQST 7.0 Ki 3
XWJGZMVWOIPRDB 7.0 Ki 4
QJNHUFOFEMCMGR 7.0 Ki 4
ARUHNEJEVKQAPD 7.0 Ki 2
BKOKSJAQZJNVPN 7.0 Ki 2
DIJNMZDNCSWBBP 7.0 Ki 2
GBNKGLWEDJOYBL 7.0 IC50 4
GWLLBXXULRHZRY 7.0 IC50 2
GWLLBXXULRHZRY 7.0 IC50 2
NRTPJMXYAMIJHJ 7.0 IC50 5
RAPDHNBJGHCCBN 7.0 Ki 3
VCHDSLCNSXYYJG 7.0 IC50 5
VGQFBYXDHFTAHX 7.0 Ki 6
VQQKGVYMJPVDSD 7.0 IC50 2
YXXOMQLSCCTIBA 7.0 Ki 4
FEAFEDHUTJTGEV 6.9 IC50 2
JGROXKKMPXLGHO 6.9 Ki 3
JVDKHRYLSLCTBR 6.9 Ki 2
NDTNHGKZDUSWEQ 6.9 Ki 4
NQEZOAWZPBBAGJ 6.9 Ki 3
PFQAPMQWNKBPIC 6.9 IC50 2
PGUPEOWWTCYVPK 6.9 Ki 4
PTCHEYWURWFAME 6.9 Ki 5
VBKUOMYCYPUADB 6.9 Ki 3
XNRMQSNQFCESPA 6.9 IC50 3
YBSXFYTXULBNOE 6.9 Ki 6
YDSJBCIWSUNWBS 6.9 Ki 2
YPBQWYRTPLXSAK 6.9 Ki 2
NEQGCINBAXAQKD 6.9 IC50 5
LWOQSODVGCORTJ 6.9 IC50 2
RKLBLCDJBJDJCD 6.9 IC50 2
VQQKGVYMJPVDSD 6.9 IC50 2
ZKPMPXGSEXIYPL 6.9 Ki 2
BGSMHNHLTFKRFT 6.9 Ki 2
KWERQAONXGOPNU 6.9 IC50 2
KWXHTGARBNTADQ 6.9 Ki 2
LLZNZOUKCHIYKS 6.9 IC50 2
LUFLMQPOYZXEPI 6.9 Ki 2
NOYRWJIVJOFKPY 6.9 IC50 2
NTNRVRBIIZBTBR 6.9 IC50 8
OHKPUUFGEUCTFI 6.9 Ki 3
QJVPWUIKUDMGJM 6.9 Ki 6
VACRFYDEAFTWGB 6.9 IC50 4
VLBYXUBKMAZVDQ 6.9 IC50 2
WLRAVKVAWRRKIZ 6.9 Ki 2
XMCSISQZUOPFCX 6.9 IC50 2
ZVOWPSKZGNRGNT 6.9 IC50 2
FRAYXFXHPHNXPH 6.9 IC50 2
2D structure