Target Details
UniProt ACP00734
Gene SymbolF2
Protein NameProthrombin
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00594 (Gla) PF00051 (Kringle) PF09396 (Thrombin_light) PF00089 (Trypsin)
Summary
  • Multi-target molecules 1,259
  • Clinical molecules 4
  • Avg pChEMBL 7.37
Top Co-occurrence Targets
Active Molecules (1,259)
InChIKey pChEMBL Type Targets Clinical
REKBLSLNDZXMEV 7.3 IC50 5
RHEKWNPDSIWZKZ 7.3 IC50 8
RXGWTRRHEHZYJO 7.3 IC50 5
SBSZVKMEHYGLPD 7.3 Ki 3
ZLJCFXPKCSWCGG 7.3 Ki 4
FPYOOPDUUPDBNP 7.3 Ki 3
JYJDBVCYQJCOFY 7.3 Ki 2
POSTYOWAJZBEMF 7.3 IC50 4
JFPVABWUQNRDDL 7.3 Ki 4
JRJYGGVSLMZUHU 7.3 IC50 3
AHBGDSREPWVVFA 7.3 IC50 2
GIQUSRUOIKSAJD 7.3 IC50 4
PLAJAOHXCUUQEL 7.3 IC50 4
PXOANDCKEAOVJN 7.3 Ki 3
BUIUMQPEDCQMFD 7.2 IC50 5
JGWDHQYXTFQAIW 7.2 IC50 2
XIBQTLNUGOHWIX 7.2 Ki 3
DZGOQOXWBUEYTK 7.2 IC50 2
GOBFKUOZUDEDMD 7.2 IC50 2
SNBIFZWZJIQRJQ 7.2 Ki 2
DFRIQJHMGZBFOM 7.2 Ki 2
YZZSRMCQLWIQSL 7.2 Ki 2
OMVUFZZIZMFUEH 7.2 Ki 2
RFEXMZCPQGEUSL 7.2 Ki 2
YVPSRJBNOKCMAX 7.2 Ki 2
RSIRPNPAPRYLFZ 7.2 IC50 4
OPEFANHGJWQXDF 7.2 IC50 4
PEWZOLRZXLOXMI 7.2 Ki 2
QPWHQTWCVWZMSE 7.2 IC50 2
YLPFNSPUPARBLY 7.2 IC50 3
PAHLSHHSYZMZRN 7.2 Ki 3
PMTJJQWYMMZALA 7.2 Ki 3
GTYRDHOPZLWHCA 7.2 IC50 3
MISMYWWUBAHTJK 7.2 Ki 4
PXVSKSKOTDZVPH 7.2 Ki 4
QQRORDHWBPBFPB 7.2 Ki 2
ZAXKLHPTMZESOW 7.2 IC50 5
HTDWCKNOXARIND 7.2 Ki 3
HTIXLULNBZFLJX 7.2 Ki 5
IPDYXCBKGJWHOF 7.2 Ki 2
JHMLZMRJAKCEAM 7.2 IC50 5
JRJYGGVSLMZUHU 7.2 IC50 2
KZFKAYHQURWCNL 7.2 Ki 2
BABFXZTUINNAIF 7.1 Ki 2
IYGMCUZMVSMAMD 7.1 IC50 2
JYGJKZKLNWLLRD 7.1 IC50 2
PGIXYPNBNAOYHW 7.1 IC50 5
VGFDMPDZPNMFII 7.1 IC50 4
FMEJXWSFZAAYQP 7.1 Ki 3
OBEJFOHWQWJNIL 7.1 Ki 7
2D structure