Target Details
| UniProt AC | P00734 |
|---|---|
| Gene Symbol | F2 |
| Protein Name | Prothrombin |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00594 (Gla) PF00051 (Kringle) PF09396 (Thrombin_light) PF00089 (Trypsin) |
Summary
- Multi-target molecules 1,259
- Clinical molecules 4
- Avg pChEMBL 7.37
KEGG Pathways (8)
Associated Diseases (2)
Active Molecules (1,259)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QZKOOEFIMWKZPK
|
7.6 | Ki | 9 | — | |
RMVFYPMRRGCHJM
|
7.6 | IC50 | 4 | — | |
SWDKZGZHCMKCKA
|
7.6 | IC50 | 2 | — | |
GBTPSLPMUMGGLO
|
7.6 | IC50 | 2 | — | |
KZNJHGCVFBGYGX
|
7.6 | Ki | 2 | — | |
RZCOAAMJHKLYHQ
|
7.6 | IC50 | 2 | — | |
VVFLUHKCTNQCLU
|
7.6 | Ki | 4 | — | |
ZRXWJXATIKDMQH
|
7.6 | IC50 | 2 | — | |
CXAXQTROOVVLBS
|
7.6 | IC50 | 2 | — | |
QAKFODQDXWPAJO
|
7.6 | Ki | 2 | — | |
QJVPFNRNEFGXGC
|
7.6 | IC50 | 2 | — | |
RXNQZXMCKASXGL
|
7.6 | IC50 | 4 | — | |
JLNIRPLGKIIBBC
|
7.6 | IC50 | 2 | — | |
CANZBHVBEWKJFW
|
7.6 | IC50 | 2 | — | |
NCBXGBVDHSJXGK
|
7.6 | IC50 | 2 | — | |
CXZHQWBVEDJXCG
|
7.6 | IC50 | 2 | — | |
GLZIACYLPINALG
|
7.6 | IC50 | 2 | — | |
KRCPVLWZQMKRME
|
7.6 | IC50 | 3 | — | |
LOMJHEAYYYPWDO
|
7.6 | IC50 | 2 | — | |
MLVTZWQEWUGCSC
|
7.6 | Ki | 5 | — | |
WYNLVLPLLLZQBA
|
7.6 | IC50 | 2 | — | |
YDLUCTVUUDEGBX
|
7.6 | IC50 | 2 | — | |
BFXKZYUODLSNBX
|
7.5 | IC50 | 2 | — | |
GJAVWABPSVJBPB
|
7.5 | Ki | 2 | — | |
JLNWZEIIEIIPES
|
7.5 | IC50 | 4 | — | |
MYYPVSMRQLUUCW
|
7.5 | IC50 | 3 | — | |
SBAHBPUZCJUMPW
|
7.5 | IC50 | 2 | — | |
WIJXQXSKKBTTEU
|
7.5 | IC50 | 2 | — | |
YJSGXHVKZSSCKV
|
7.5 | IC50 | 2 | — | |
ZJDGGFCBBONCDM
|
7.5 | IC50 | 2 | — | |
DBLNNDOSJLJNTF
|
7.5 | Ki | 4 | — | |
FYBMKIHEKBWKGO
|
7.5 | Ki | 2 | — | |
HTOGBQJUJBBWIE
|
7.5 | Ki | 4 | — | |
UPWRYEAGKLIQQY
|
7.5 | IC50 | 2 | — | |
HECONMODEBIAKY
|
7.5 | IC50 | 9 | — | |
KTWUUUQCPDYETH
|
7.5 | Ki | 2 | — | |
OBRCAKGVHQFHGX
|
7.5 | Ki | 4 | — | |
UNTYULOIKNKYHN
|
7.5 | IC50 | 3 | — | |
SGWQBTZXXBLNJR
|
7.5 | IC50 | 2 | — | |
HCONWOFFAXZHQA
|
7.5 | Ki | 4 | — | |
HRGKDTRCXPZMHG
|
7.5 | IC50 | 2 | — | |
LOITXWAIWLBDGR
|
7.5 | Ki | 2 | — | |
OOSFXPQKGFCWRC
|
7.5 | IC50 | 7 | — | |
MWJAQZALXIOOQS
|
7.5 | Ki | 2 | — | |
QBIQHSJYZKKJPJ
|
7.5 | Ki | 4 | — | |
UZMQVFWUMDZRLA
|
7.5 | Ki | 2 | — | |
BVIZJIXKCBABFU
|
7.5 | IC50 | 4 | — | |
JBAZPOYGAUQDAO
|
7.5 | Ki | 2 | — | |
BOWCZWCYXWJVHD
|
7.5 | Ki | 3 | — | |
DFRIQJHMGZBFOM
|
7.5 | Ki | 2 | — |