Target Details
UniProt ACP00734
Gene SymbolF2
Protein NameProthrombin
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00594 (Gla) PF00051 (Kringle) PF09396 (Thrombin_light) PF00089 (Trypsin)
Summary
  • Multi-target molecules 1,259
  • Clinical molecules 4
  • Avg pChEMBL 7.37
Top Co-occurrence Targets
Active Molecules (1,259)
InChIKey pChEMBL Type Targets Clinical
FSVAWWOYUSROJH 11.6 Ki 3
SJIGBLXECWIEFM 11.5 Ki 2
WJVLTXKAUHPMNM 11.5 Ki 2
CRPPBRFZGAUWJM 11.3 Ki 2
IHBRTJZRICMSLW 11.1 IC50 4
MQPQHCSONVFZIT 10.9 Ki 2
OPOYAWWWOKBVEB 10.8 Ki 6
BIHPYGVYKSQDLA 10.8 Ki 6
DLEWBCCCSUQVHV 10.7 Ki 4
VHDSIUDQBOQQLE 10.7 Ki 2
PWVZGBVCDDZZNQ 10.7 Ki 3
UQMOAGGBXALCSZ 10.7 Ki 2
GOBXSXIHPUGHDS 10.6 Ki 6
WTMZVIILZZXXFO 10.5 Ki 2
MERYTOPZZMIEFD 10.5 Ki 3
CDJAIRYCIJZATA 10.4 Ki 6
FXFYPTZERULUBS 10.4 Ki 3
MPSGQHXXALMTIC 10.4 Ki 2
NNTAUPYRIUVLBN 10.4 Ki 2
FXFYPTZERULUBS 10.4 Ki 5
OWCMVQFLPIOYNL 10.4 Ki 4
QPBFLOWZPFHTHE 10.4 Ki 6
DKHWNGVLBHNOLG 10.3 Ki 3
FXFYPTZERULUBS 10.3 Ki 3
BKMLZHDSJSJXNS 10.3 Ki 3
GDGNUENLKMKSGL 10.3 Ki 2
SFGQHQOPLLWNCX 10.3 Ki 3
SYJMIXHRYXUAGD 10.2 Ki 2
AHVRHIQTLPAZHX 10.2 Ki 2
DCUODGWOKBGFJV 10.2 Ki 3
DSVGBRXCGKCTSK 10.2 Ki 2
KEWCBOBJEQHYIV 10.2 Ki 6
UNIOGIZCWAGOKV 10.2 Ki 6
VQXMYKHZVHNFTJ 10.2 Ki 4
AYWIUHKKDARFIP 10.1 Ki 2
LYVSCNRRXJZCRV 10.1 Ki 2
MHZINYCTUDNOIC 10.0 Ki 3
OECPVFSZEWVKDZ 10.0 Ki 2
OYGPPOOTDFYCCI 10.0 Ki 2
SEBIKUOIXHBWMY 10.0 Ki 2
ZAXAEIBEVRYJIB 10.0 IC50 2
FNTHJTUPRVAXFZ 10.0 IC50 17
XMSAWCPABLSFFM 10.0 Ki 6
DJNNZKJZFCRFRX 10.0 Ki 4
FDCBFBSFHLWFFU 10.0 Ki 6
RBXLABNLPAAXCE 9.9 Ki 2
AJEASRLDZKLAGW 9.9 Ki 2
SAHIWIHDGKJMDR 9.9 Ki 5
ANKIJLVYTUKGJM 9.8 Ki 6
QTGRXIGBXXVLEH 9.8 Ki 3
2D structure