Target Details
| UniProt AC | P00521 |
|---|---|
| Gene Symbol | ABL |
| Protein Name | Tyrosine-protein kinase transforming protein Abl |
| Organism | Abelson murine leukemia virus |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF08919 (F_actin_bind) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) |
Summary
- Multi-target molecules 5
- Clinical molecules 5
- Avg pChEMBL 6.81
Active Molecules (5)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LSPANGZZENHZNJ
|
7.5 | IC50 | 10 | Yes | |
DBDQLLPCPIODHI
|
6.8 | IC50 | 5 | Yes | |
DVMBLTDKHALLLH
|
6.7 | IC50 | 6 | Yes | |
BUGPWXMPCMTLIX
|
6.6 | IC50 | 7 | Yes | |
ZDNMTYMNWKRHQA
|
6.4 | IC50 | 5 | Yes |