Target Details
| UniProt AC | P00519 |
|---|---|
| Gene Symbol | ABL1 |
| Protein Name | Tyrosine-protein kinase ABL1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08919 (F_actin_bind) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,419
- Clinical molecules 468
- Avg pChEMBL 7.25
KEGG Pathways (12)
Associated Diseases (3)
Active Molecules (1,419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GMYQHOQOEQWZGN
|
7.6 | IC50 | 3 | — | |
HRRMXIICSWVXIS
|
7.6 | IC50 | 13 | Yes | |
MPYUMMWCLQVMLG
|
7.6 | IC50 | 11 | — | |
VAPRWSMRTJIVDQ
|
7.6 | IC50 | 4 | — | |
BLYRPGBSIKAIAU
|
7.6 | IC50 | 24 | Yes | |
FSFYBWMHVKFOOV
|
7.6 | IC50 | 5 | — | |
IWGLXKVBQSBQMC
|
7.6 | IC50 | 13 | Yes | |
JBPBNXCKEHXPOS
|
7.6 | IC50 | 2 | — | |
MLSMCXWBTQUJBM
|
7.6 | IC50 | 2 | — | |
SFYPWBCTUYQPBH
|
7.6 | Ki | 2 | — | |
UNBNKYSPLOMIOY
|
7.6 | IC50 | 7 | — | |
AQPGSKXVUOGJPP
|
7.6 | IC50 | 2 | — | |
BNIPBKFCGMYCDD
|
7.6 | IC50 | 2 | — | |
MULNSLQVKKUPJN
|
7.6 | Ki | 41 | — | |
QHXBWJSQXSYAGG
|
7.6 | IC50 | 16 | — | |
WJEOLQLKVOPQFV
|
7.6 | Kd | 24 | — | |
XKFTZKGMDDZMJI
|
7.6 | IC50 | 8 | Yes | |
ZGDSBEUMPIMXBM
|
7.6 | Ki | 42 | — | |
DOVNUEPFPBWTSV
|
7.6 | IC50 | 2 | — | |
IQIXKGNNKIOWHL
|
7.6 | IC50 | 2 | — | |
OMVOXDNRIIIPHG
|
7.6 | IC50 | 2 | — | |
QYPSALIXKCRYNZ
|
7.6 | IC50 | 12 | Yes | |
SQJDLYFEJSIHPR
|
7.6 | IC50 | 2 | — | |
XESOUPPNAWVWAG
|
7.6 | IC50 | 2 | — | |
ZTQOHJNXDAUMOA
|
7.6 | IC50 | 13 | Yes | |
ZWEHYQSGMOUIRZ
|
7.6 | Ki | 3 | — | |
LXRITECWUGVGTD
|
7.6 | IC50 | 6 | — | |
RVVOZOVEPBDKNY
|
7.6 | IC50 | 2 | — | |
GUEFRZZGCQAGLR
|
7.5 | IC50 | 2 | — | |
RTRHXDLGBINMNM
|
7.5 | IC50 | 5 | — | |
UVFLAWMNLLGDNC
|
7.5 | IC50 | 2 | — | |
BVQJGEBCGLWTNC
|
7.5 | IC50 | 3 | — | |
DIMLYBUSJYNUFT
|
7.5 | Kd | 6 | — | |
OWSMSMNEFKFQBZ
|
7.5 | IC50 | 3 | — | |
DBHZLVWJMDYRBG
|
7.5 | IC50 | 3 | — | |
YYLKKYCXAOBSRM
|
7.5 | Kd | 191 | — | |
JLQPVUJUCFSACM
|
7.5 | IC50 | 2 | — | |
LSPANGZZENHZNJ
|
7.5 | IC50 | 10 | Yes | |
NSRFIEYUXOOISZ
|
7.5 | IC50 | 2 | — | |
OJOMKFBUCUYZRW
|
7.5 | IC50 | 3 | — | |
OUKYUETWWIPKQR
|
7.5 | IC50 | 31 | Yes | |
OZLFFPLKFGJQDT
|
7.5 | IC50 | 2 | — | |
PPRRKOMHIBJJKA
|
7.5 | IC50 | 2 | — | |
QFKVEVOGGCTCKS
|
7.5 | IC50 | 2 | — | |
SMWFHLHWOOWYAP
|
7.5 | IC50 | 4 | Yes | |
SWWHQLAUNHTMIH
|
7.5 | IC50 | 2 | — | |
UEHGHDJPDQDZPX
|
7.5 | IC50 | 3 | — | |
VFUZEFVLUHADNS
|
7.5 | IC50 | 4 | Yes | |
XJNQIRXYMVFKTA
|
7.5 | IC50 | 3 | — | |
ZLNBJDSAGVBJSP
|
7.5 | IC50 | 8 | Yes |