Target Details
| UniProt AC | P00519 |
|---|---|
| Gene Symbol | ABL1 |
| Protein Name | Tyrosine-protein kinase ABL1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08919 (F_actin_bind) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,419
- Clinical molecules 468
- Avg pChEMBL 7.25
KEGG Pathways (12)
Associated Diseases (3)
Active Molecules (1,419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NVRXTLZYXZNATH
|
7.8 | IC50 | 47 | Yes | |
TZEWBPGVTYPITP
|
7.8 | IC50 | 5 | — | |
YRDHKIFCGOZTGD
|
7.8 | IC50 | 21 | — | |
CDRJTNGWNAODES
|
7.7 | IC50 | 3 | Yes | |
CJZDHNAPSGIJPC
|
7.7 | IC50 | 2 | — | |
DITRHERLQQIVDS
|
7.7 | IC50 | 2 | — | |
FCDMJPPRJSFFRX
|
7.7 | IC50 | 2 | — | |
LHVHGXVPJPMLFB
|
7.7 | IC50 | 2 | — | |
NYKXOFIGGDPRIF
|
7.7 | IC50 | 2 | — | |
VWCSBXLDSKERLY
|
7.7 | IC50 | 2 | — | |
JRJBXDYPYRFVHH
|
7.7 | IC50 | 2 | — | |
KODAMADJHOKWQH
|
7.7 | IC50 | 2 | — | |
ONXVBFWIQSGWAH
|
7.7 | IC50 | 2 | — | |
QMWCOMCAODPOMZ
|
7.7 | IC50 | 2 | — | |
UPZUOJCELONEIR
|
7.7 | IC50 | 2 | — | |
WPSWNDSKLXFMIS
|
7.7 | IC50 | 2 | — | |
YJQOQJNKFYBZOV
|
7.7 | IC50 | 2 | — | |
OTTCBLPTHPBEEX
|
7.7 | Ki | 11 | Yes | |
PELIWNRKLAFPFO
|
7.7 | IC50 | 2 | — | |
AFVGAHBUCVDPPI
|
7.7 | IC50 | 6 | Yes | |
CGECJCJUHCZZGO
|
7.7 | IC50 | 9 | — | |
MFDCEMLTTQCDTH
|
7.7 | IC50 | 3 | Yes | |
PPHMKXKASWTCSZ
|
7.7 | IC50 | 2 | Yes | |
QPEWSVDGDKWHMX
|
7.7 | IC50 | 2 | — | |
YKDNQUNPTIJKCH
|
7.7 | IC50 | 2 | — | |
FAXUBOMVBMGLNX
|
7.7 | IC50 | 2 | — | |
CBMGZXHASOIHSW
|
7.7 | IC50 | 2 | — | |
COAQRADEUYYCDG
|
7.7 | IC50 | 12 | Yes | |
CYYRPFWAMVGRGT
|
7.7 | IC50 | 3 | — | |
HHZIURLSWUIHRB
|
7.7 | IC50 | 57 | Yes | |
MRZVUZUMBCEAGI
|
7.7 | IC50 | 12 | Yes | |
MRZVUZUMBCEAGI
|
7.7 | IC50 | 11 | Yes | |
QNKRFRCYRMDLLE
|
7.7 | Ki | 2 | — | |
RZKBSKVRXHFGJG
|
7.7 | IC50 | 3 | — | |
SWYGYHUKYVHTHP
|
7.7 | IC50 | 2 | — | |
YZMSPABNYFHEHD
|
7.7 | IC50 | 2 | — | |
YZRLWPBYTMKRQR
|
7.7 | IC50 | 11 | — | |
ZSHRAUSJZQDIJR
|
7.7 | IC50 | 9 | Yes | |
BMFUIUDLVMJYGT
|
7.7 | IC50 | 3 | — | |
JXYHYYBXKLTNGG
|
7.7 | IC50 | 3 | — | |
KVTMDRDZMBVWNC
|
7.7 | IC50 | 6 | — | |
AZTXEXSCWBYKOB
|
7.7 | IC50 | 2 | — | |
CEUSZLVORFRBCV
|
7.7 | IC50 | 13 | — | |
GMHHKAPVIOBKKS
|
7.7 | IC50 | 2 | — | |
KTTGLAHMSDMRLJ
|
7.7 | IC50 | 12 | Yes | |
LZYWVOKHWFMDJU
|
7.7 | IC50 | 3 | — | |
MGSXHFUDTNNPGZ
|
7.7 | IC50 | 2 | — | |
SQXJLEVGNHLDCC
|
7.7 | IC50 | 6 | Yes | |
ZDNURMVOKAERHZ
|
7.7 | IC50 | 7 | Yes | |
MIARGORLLRWINC
|
7.7 | IC50 | 2 | — |