Target Details
| UniProt AC | P00519 |
|---|---|
| Gene Symbol | ABL1 |
| Protein Name | Tyrosine-protein kinase ABL1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08919 (F_actin_bind) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,419
- Clinical molecules 468
- Avg pChEMBL 7.25
KEGG Pathways (12)
Associated Diseases (3)
Active Molecules (1,419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BWLSIYJKVFXNFV
|
7.9 | IC50 | 4 | Yes | |
JXVHQHBMOSSYBX
|
7.9 | IC50 | 3 | — | |
UDRCHZMTVKQTAE
|
7.9 | IC50 | 3 | — | |
WPHKIQPVPYJNAX
|
7.9 | IC50 | 81 | — | |
ZGBAJMQHJDFTQJ
|
7.9 | IC50 | 15 | — | |
ZGBAJMQHJDFTQJ
|
7.9 | IC50 | 2 | — | |
CQCOXFUOMTWNCR
|
7.9 | IC50 | 2 | — | |
MJZHYLCYHDBDFA
|
7.9 | IC50 | 2 | — | |
PELIWNRKLAFPFO
|
7.9 | IC50 | 2 | — | |
UQNNJYLAPYGZBD
|
7.9 | Ki | 28 | — | |
AWIQZKGARNWZPQ
|
7.9 | IC50 | 2 | — | |
GCIKSSRWRFVXBI
|
7.9 | Kd | 109 | Yes | |
MWUBHDHHMFIRMG
|
7.9 | IC50 | 2 | — | |
NEHHEDJQRHQOOW
|
7.9 | IC50 | 5 | — | |
OKPRPWYLQUKXFE
|
7.9 | IC50 | 7 | Yes | |
SAYPRYYFORNPCK
|
7.9 | IC50 | 2 | — | |
FVYMRGNWPDZIDO
|
7.9 | IC50 | 2 | — | |
SVYYVGZMWJYFIE
|
7.9 | IC50 | 3 | — | |
PELIWNRKLAFPFO
|
7.9 | IC50 | 2 | — | |
ALKJNCZNEOTEMP
|
7.8 | IC50 | 55 | — | |
CJMMCIXRPVLDBH
|
7.8 | IC50 | 12 | Yes | |
IHYVCWMRZWUYDY
|
7.8 | IC50 | 2 | — | |
MGQBHVRGZCUQID
|
7.8 | IC50 | 2 | — | |
HYMHVNNHIASECU
|
7.8 | IC50 | 5 | — | |
TWUHJIAGJSKONL
|
7.8 | IC50 | 2 | — | |
GMTZLHADUFDDDN
|
7.8 | IC50 | 5 | — | |
ZGJPEVGMGPUSJY
|
7.8 | IC50 | 2 | — | |
ABIOEYXBRUITSN
|
7.8 | IC50 | 2 | — | |
VASBUQQNBORQFF
|
7.8 | IC50 | 2 | — | |
WBVZVKAMQLVYTF
|
7.8 | IC50 | 2 | — | |
WHTLLTQCEBVRBM
|
7.8 | IC50 | 2 | — | |
FSHQMSATUUIMTE
|
7.8 | Ki | 3 | Yes | |
HHOVYYSFRMBKPP
|
7.8 | IC50 | 3 | Yes | |
KCPUHXYDPHVBQZ
|
7.8 | IC50 | 2 | — | |
LAVCQCXXKFSGQN
|
7.8 | IC50 | 2 | — | |
ONVKFNZGEFTWQD
|
7.8 | IC50 | 4 | Yes | |
UOOZSMNSBYVUGZ
|
7.8 | Ki | 32 | — | |
ZIXANSQHENONFN
|
7.8 | IC50 | 2 | — | |
LDGJWNZFGYFENB
|
7.8 | IC50 | 2 | — | |
COAQRADEUYYCDG
|
7.8 | IC50 | 12 | Yes | |
DECSMGXZYHHMMF
|
7.8 | IC50 | 2 | — | |
NKEZCSVNPKYVIB
|
7.8 | IC50 | 2 | — | |
RONIOIPFUMELRH
|
7.8 | IC50 | 4 | Yes | |
SUNRRXUOOBKXTB
|
7.8 | IC50 | 2 | — | |
BJCJYEYYYGBROF
|
7.8 | IC50 | 4 | — | |
PITUMGJELDUJEZ
|
7.8 | IC50 | 3 | Yes | |
QOKBZTDZIZMTMS
|
7.8 | IC50 | 2 | — | |
AZOXWOCICFEBCQ
|
7.8 | IC50 | 11 | — | |
CDXRBIMKCWWDMY
|
7.8 | IC50 | 2 | — | |
FOYDGOBFRZQHEU
|
7.8 | IC50 | 13 | — |