Target Details
| UniProt AC | P00519 |
|---|---|
| Gene Symbol | ABL1 |
| Protein Name | Tyrosine-protein kinase ABL1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08919 (F_actin_bind) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,419
- Clinical molecules 468
- Avg pChEMBL 7.25
KEGG Pathways (12)
Associated Diseases (3)
Active Molecules (1,419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BDHJKYLJPYEWOX
|
8.1 | IC50 | 2 | — | |
DMWAXJBYXJFYAH
|
8.1 | IC50 | 2 | — | |
HMWBDNPYGWPLRR
|
8.1 | IC50 | 2 | Yes | |
PELIWNRKLAFPFO
|
8.1 | IC50 | 3 | — | |
PJGIZSKNZNTQMF
|
8.1 | IC50 | 2 | — | |
XOVYHZSDUHWRJV
|
8.1 | IC50 | 6 | Yes | |
BXUFOTJKNXPVHP
|
8.1 | Ki | 2 | — | |
FEYMWTKZTZABTA
|
8.1 | IC50 | 2 | — | |
HFGDXJQGICLTIE
|
8.1 | IC50 | 5 | — | |
KUNZDWIFPOMUOX
|
8.1 | Ki | 36 | — | |
MNBNPSZPKJMKII
|
8.1 | IC50 | 2 | — | |
OWRXHGAFWZFFCW
|
8.1 | Ki | 113 | — | |
RKGOHOXKHIGYOL
|
8.1 | IC50 | 2 | — | |
RTYJMUXLFRYRBU
|
8.1 | Ki | 35 | — | |
XKFTZKGMDDZMJI
|
8.1 | IC50 | 64 | Yes | |
HTZNZEKPDCTESZ
|
8.1 | IC50 | 6 | Yes | |
MYMBTVRXCNFFNP
|
8.1 | IC50 | 2 | — | |
YAFBWUKWKZZPIF
|
8.1 | IC50 | 4 | Yes | |
YQWRDEHPSFGGHV
|
8.1 | IC50 | 4 | Yes | |
RCMBBRKIGQGXGS
|
8.1 | IC50 | 2 | — | |
REKRJPDVODUIMJ
|
8.1 | IC50 | 2 | — | |
HQXLJEBXFZNYOC
|
8.1 | IC50 | 2 | — | |
LCMCFIMDFHOMQO
|
8.1 | IC50 | 2 | — | |
RGDCBCQGGRTXNW
|
8.1 | IC50 | 2 | — | |
HJALCEUIPSPHHD
|
8.0 | IC50 | 2 | — | |
PLZOWXHKTJJSQR
|
8.0 | IC50 | 3 | Yes | |
WAFBXGBWFZZGIC
|
8.0 | IC50 | 3 | — | |
KQOYBUCRLZDLBE
|
8.0 | IC50 | 3 | — | |
ZWVLMQTXUWMUII
|
8.0 | IC50 | 9 | Yes | |
YDELNSXADYPQGS
|
8.0 | IC50 | 15 | Yes | |
AUTOLBMXDDTRRT
|
8.0 | IC50 | 3 | — | |
CGMQSJXTBXHOTH
|
8.0 | IC50 | 9 | — | |
DPSNOZFUMXEANO
|
8.0 | Kd | 7 | — | |
GKDGNKRGOJPYMM
|
8.0 | IC50 | 2 | — | |
KKYPRNBBPBRJQX
|
8.0 | Ki | 40 | — | |
KOHNRDPXFDZZJF
|
8.0 | Ki | 31 | — | |
NRSRGKSRBDKZAU
|
8.0 | IC50 | 2 | — | |
ODPGGGTTYSGTGO
|
8.0 | Kd | 153 | — | |
SBLMCLDRWJNEJK
|
8.0 | IC50 | 17 | — | |
TVUWQDLBEOZVOU
|
8.0 | Ki | 41 | — | |
TWGQYAXRDILACQ
|
8.0 | IC50 | 2 | — | |
UUWNXFJBBYAMDT
|
8.0 | Ki | 46 | — | |
WXLDRYNTEQUKFN
|
8.0 | IC50 | 2 | — | |
KUNOALCWXLLCES
|
8.0 | IC50 | 2 | — | |
LWGSLBQDPISOIG
|
8.0 | IC50 | 2 | — | |
RZHUMJSINYZTBK
|
8.0 | IC50 | 2 | — | |
YJSFAHMGDRBZGH
|
8.0 | Ki | 16 | Yes | |
YFYPWCVYZUWOGM
|
8.0 | IC50 | 2 | — | |
AMHUBFWCCMLLCJ
|
7.9 | IC50 | 15 | — | |
APGJWCRRERWKDQ
|
7.9 | IC50 | 6 | Yes |