Target Details
| UniProt AC | P00519 |
|---|---|
| Gene Symbol | ABL1 |
| Protein Name | Tyrosine-protein kinase ABL1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08919 (F_actin_bind) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,419
- Clinical molecules 468
- Avg pChEMBL 7.25
KEGG Pathways (12)
Associated Diseases (3)
Active Molecules (1,419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NMSHJWKGPWRUSI
|
8.4 | Ki | 2 | — | |
YIUOPZRKRRRSTC
|
8.4 | IC50 | 2 | — | |
INSVCYRFDCTMIA
|
8.4 | IC50 | 5 | — | |
PQRFMBAACAPZPP
|
8.4 | IC50 | 12 | Yes | |
UMBIRSZUCJNBHB
|
8.4 | IC50 | 18 | — | |
ZCWRJICNHZNBPI
|
8.4 | IC50 | 2 | — | |
PDEWZRGITAXNMH
|
8.4 | Ki | 2 | — | |
FNEDDGRJWXWDNZ
|
8.3 | IC50 | 5 | — | |
MXWHSGSOZDOVLL
|
8.3 | IC50 | 4 | Yes | |
ZLMVXCGWUJXFNP
|
8.3 | IC50 | 15 | Yes | |
BYRBUVTUGSOTSC
|
8.3 | IC50 | 7 | Yes | |
HRJNCGVLSVNXDX
|
8.3 | IC50 | 2 | — | |
KWLXWXYINQHVEA
|
8.3 | IC50 | 2 | — | |
TUXQTYDDHNAJKZ
|
8.3 | IC50 | 6 | Yes | |
XWTBASUJPOEBBZ
|
8.3 | IC50 | 6 | Yes | |
GNIYUURCQFKRCB
|
8.3 | IC50 | 11 | Yes | |
JKDJAOQUTMBBQB
|
8.3 | IC50 | 5 | — | |
KEIRBRQKXFLPHS
|
8.3 | IC50 | 3 | — | |
PYGLWXFBTJNWSQ
|
8.3 | Ki | 2 | — | |
WQACVRFKZIYHIM
|
8.3 | Ki | 3 | Yes | |
XCIWPOBMQAYXJN
|
8.3 | IC50 | 6 | Yes | |
ZUMNLSFJINJANM
|
8.3 | IC50 | 5 | Yes | |
PUJPRSYMMNNGBM
|
8.3 | Ki | 2 | — | |
DJCLBOJZORFUMR
|
8.3 | IC50 | 2 | — | |
IQOAIXAFDYRGNK
|
8.3 | IC50 | 3 | — | |
XLLINEQPLUTYIF
|
8.3 | IC50 | 7 | Yes | |
PZINVJUNZRLUIM
|
8.3 | IC50 | 3 | — | |
ZBTLTVIYBHYEHL
|
8.3 | IC50 | 13 | Yes | |
PCSKFQHKWWNIKM
|
8.2 | IC50 | 7 | — | |
KIHQVERTLRHJED
|
8.2 | IC50 | 2 | — | |
WDNAXOPVZIEECR
|
8.2 | IC50 | 11 | — | |
XVJQXIUEEXVEKU
|
8.2 | IC50 | 3 | — | |
FVOSLYACENHGIN
|
8.2 | IC50 | 2 | — | |
IUCMEDMSUCVZQN
|
8.2 | IC50 | 2 | — | |
MAEHWTXHQDRFIE
|
8.2 | IC50 | 2 | — | |
ROHJEIACUNTGFP
|
8.2 | IC50 | 16 | — | |
SZPKERXOPUWUPW
|
8.2 | IC50 | 3 | — | |
JVGNHFZOVWJKER
|
8.2 | IC50 | 3 | — | |
WQERLKAGPFFGAY
|
8.2 | IC50 | 2 | — | |
MBPKPSDAPFPECJ
|
8.2 | IC50 | 12 | Yes | |
GCDSDVNITVBCDW
|
8.2 | IC50 | 17 | — | |
IZPYRHJDUKTQPR
|
8.2 | IC50 | 2 | — | |
KMMUTXPSVYLUNZ
|
8.2 | IC50 | 3 | — | |
ZCQBIMLCHPNRKB
|
8.2 | IC50 | 3 | — | |
LHZOGDYGAMOXIH
|
8.2 | IC50 | 2 | Yes | |
QKKIWEILHCXECO
|
8.2 | IC50 | 24 | — | |
CNTAQWMENZCDOK
|
8.2 | IC50 | 2 | — | |
FQXQXOYNTXHBKK
|
8.2 | IC50 | 7 | — | |
GKVWMMLQQGMAMC
|
8.2 | IC50 | 2 | — | |
AKFZSHPZKXBMCK
|
8.1 | IC50 | 2 | — |