Target Details
| UniProt AC | P00519 |
|---|---|
| Gene Symbol | ABL1 |
| Protein Name | Tyrosine-protein kinase ABL1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08919 (F_actin_bind) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,419
- Clinical molecules 468
- Avg pChEMBL 7.25
KEGG Pathways (12)
Associated Diseases (3)
Active Molecules (1,419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XKFTZKGMDDZMJI
|
8.6 | Ki | 56 | — | |
XKZINYYXWJEYEL
|
8.6 | Ki | 37 | — | |
XOOAAYRIVATZNM
|
8.6 | Ki | 55 | — | |
XVCPZFLMAOLHQX
|
8.6 | IC50 | 2 | — | |
YLOVBNCIDYKIDW
|
8.6 | IC50 | 8 | Yes | |
DFQQSYDMGWRPAN
|
8.6 | IC50 | 3 | — | |
XKCPEVHEMILVAL
|
8.6 | IC50 | 2 | — | |
MLLBPOJSIGXWLG
|
8.6 | IC50 | 3 | Yes | |
YIUOPZRKRRRSTC
|
8.6 | IC50 | 2 | — | |
WVXNSAVVKYZVOE
|
8.6 | IC50 | 92 | — | |
ZIQFYVPVJZEOFS
|
8.6 | IC50 | 9 | Yes | |
FCIILWHQWNLPJU
|
8.5 | IC50 | 4 | Yes | |
FHUDMNMPUCFLRX
|
8.5 | IC50 | 2 | — | |
HJVDQPRJANOXIX
|
8.5 | IC50 | 10 | — | |
KDTFQAJYJIGSFS
|
8.5 | Ki | 2 | — | |
QXIOZIFTPMAING
|
8.5 | IC50 | 17 | — | |
TXAYKQMEBQBGLR
|
8.5 | IC50 | 4 | Yes | |
DKNUPRMJNUQNHR
|
8.5 | Kd | 33 | — | |
VWBZVMZFOBZQTD
|
8.5 | IC50 | 2 | Yes | |
WFRLFWGASBLYTC
|
8.5 | IC50 | 15 | Yes | |
ZBRROTSBDAODQD
|
8.5 | Ki | 7 | Yes | |
YIUOPZRKRRRSTC
|
8.5 | IC50 | 2 | — | |
ADLPKFFMGIJZIM
|
8.5 | Ki | 44 | — | |
RITAVMQDGBJQJZ
|
8.5 | Ki | 33 | — | |
KOGBNTSOPZVMIK
|
8.5 | IC50 | 2 | — | |
SCVOABYBOHRDLK
|
8.5 | IC50 | 2 | — | |
AIKGYQDFIJRQIY
|
8.5 | IC50 | 9 | — | |
DOBZFFWLHXORTB
|
8.5 | Ki | 2 | — | |
DQLDULIEUKHCJI
|
8.5 | Ki | 2 | — | |
YIUOPZRKRRRSTC
|
8.5 | IC50 | 2 | — | |
GPTPEUDRFUOZSX
|
8.5 | Ki | 2 | — | |
VZSXRPCZRQJQFY
|
8.5 | Ki | 2 | — | |
CLVFHIUJCJCESW
|
8.5 | IC50 | 2 | — | |
HXVYZZYPRMCJGZ
|
8.5 | IC50 | 2 | — | |
VAWLAPYBUJTXRS
|
8.5 | Ki | 6 | Yes | |
ZPKGDYKWVKCDJQ
|
8.5 | IC50 | 4 | Yes | |
KNXQEJUJQOZAKP
|
8.4 | IC50 | 7 | Yes | |
RFSFIDGEFVXSQM
|
8.4 | IC50 | 12 | Yes | |
SYZNYVDAHCWNHN
|
8.4 | IC50 | 2 | — | |
WZIXOSLCIKUWAH
|
8.4 | IC50 | 2 | — | |
SXIDXVGGABQPIG
|
8.4 | IC50 | 2 | — | |
USIPMCNVJIUSIH
|
8.4 | IC50 | 2 | — | |
RIWJSTAVOOCXPT
|
8.4 | IC50 | 3 | — | |
FDVSOQRNTAPCHB
|
8.4 | Ki | 40 | — | |
LOLPPWBBNUVNQZ
|
8.4 | IC50 | 97 | Yes | |
RBXYGQNZRVPDNB
|
8.4 | Ki | 34 | — | |
UVHMCYBDLLCIAP
|
8.4 | IC50 | 2 | — | |
YDWMUCKJUNLURC
|
8.4 | Ki | 24 | — | |
ZGBAJMQHJDFTQJ
|
8.4 | IC50 | 2 | — | |
GMCVFFUTKQUYKX
|
8.4 | IC50 | 2 | — |