Target Details
| UniProt AC | P00519 |
|---|---|
| Gene Symbol | ABL1 |
| Protein Name | Tyrosine-protein kinase ABL1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08919 (F_actin_bind) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,419
- Clinical molecules 468
- Avg pChEMBL 7.25
KEGG Pathways (12)
Associated Diseases (3)
Active Molecules (1,419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YLGBXIFLTCUQDE
|
9.0 | IC50 | 2 | — | |
GOEIHELWQGXKOI
|
9.0 | IC50 | 2 | — | |
KJOGLHQXZFOMRY
|
8.9 | IC50 | 2 | — | |
AWJZZXXWVQWGDE
|
8.9 | IC50 | 2 | — | |
DUPWHXBITIZIKZ
|
8.9 | IC50 | 2 | — | |
DZUFTTMDQLYMBE
|
8.9 | IC50 | 10 | Yes | |
FZBVNCFBCNXULH
|
8.9 | IC50 | 18 | — | |
LIEUQFMVFKJKHX
|
8.9 | Kd | 10 | — | |
UDUPSRWUDACGIS
|
8.9 | IC50 | 13 | Yes | |
VTWWRKFUHCSCEW
|
8.9 | Kd | 19 | — | |
SZNYUUZOQHNEKB
|
8.9 | IC50 | 7 | — | |
XBYVOPRDASFDMY
|
8.9 | Ki | 42 | — | |
CSXVLYGUGWXOAL
|
8.9 | Ki | 2 | — | |
IBRPSHUYWHRYQA
|
8.9 | IC50 | 4 | Yes | |
LYADGAGFYYXXIO
|
8.9 | IC50 | 82 | — | |
NHCXDULQCCCWLO
|
8.9 | IC50 | 3 | — | |
APPAUNZXIPSWAS
|
8.8 | IC50 | 7 | Yes | |
IQSSNBZGOCNVDV
|
8.8 | IC50 | 2 | — | |
KNTPBVJWLVSQOV
|
8.8 | IC50 | 2 | — | |
VAARYSWULJUGST
|
8.8 | Kd | 119 | Yes | |
KJIJJDDZGNJZBA
|
8.8 | IC50 | 2 | — | |
QAMUWRFOZKONDU
|
8.8 | IC50 | 7 | — | |
WJUMXJCIOLETKL
|
8.8 | IC50 | 2 | — | |
AQSSMEORRLJZLU
|
8.8 | Ki | 34 | Yes | |
MCCCQFAOMZMZKE
|
8.8 | Ki | 52 | — | |
NWUCBGDFEQGJTP
|
8.8 | IC50 | 2 | Yes | |
PXEXUKNUARXICD
|
8.8 | IC50 | 2 | Yes | |
QAZSOKNYSVTMPH
|
8.8 | IC50 | 3 | — | |
UGEJLCNSVIVALC
|
8.8 | Ki | 41 | — | |
VCFDMLBPASGZTP
|
8.8 | Ki | 38 | — | |
PPBMKPYHIGDXNE
|
8.8 | IC50 | 2 | — | |
BCGSHQSXJFPEKN
|
8.8 | IC50 | 2 | — | |
DNLQIFRJOZJGCU
|
8.8 | Ki | 6 | Yes | |
RCZHVXSTTOXWRM
|
8.8 | Ki | 3 | — | |
BWHGYXORZLZUIK
|
8.7 | IC50 | 2 | Yes | |
UOVRWDKWWSPLGT
|
8.7 | IC50 | 2 | — | |
BRTHUECZMVKNMQ
|
8.7 | Ki | 31 | — | |
KNACLJBHKVSTDL
|
8.7 | Ki | 40 | — | |
ULHGAQSVFPOUDY
|
8.7 | Ki | 43 | — | |
ZCCJKVBTHCOISJ
|
8.7 | Ki | 46 | — | |
URNMUIDFWOJTPW
|
8.7 | Ki | 7 | Yes | |
YTHUQGIGAIZNIM
|
8.7 | IC50 | 3 | — | |
KGUOPPORYLAEOV
|
8.7 | IC50 | 2 | — | |
NFLXEOXSZWSZGF
|
8.6 | IC50 | 2 | — | |
QSECCHMWSVTBKZ
|
8.6 | IC50 | 4 | Yes | |
XCYATSRJUCZIJR
|
8.6 | IC50 | 7 | Yes | |
IWGIXRMJMSKLGP
|
8.6 | IC50 | 4 | Yes | |
YHVHYWYQEFELOW
|
8.6 | IC50 | 44 | — | |
CIKRVGZNQZNXMQ
|
8.6 | IC50 | 2 | — | |
XJSFDMGICAWQFS
|
8.6 | Ki | 60 | — |