Target Details
| UniProt AC | P00519 |
|---|---|
| Gene Symbol | ABL1 |
| Protein Name | Tyrosine-protein kinase ABL1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08919 (F_actin_bind) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,419
- Clinical molecules 468
- Avg pChEMBL 7.25
KEGG Pathways (12)
Associated Diseases (3)
Active Molecules (1,419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BPQBMWJXOIQOCG
|
9.3 | IC50 | 3 | — | |
DKNHELJFXSXKQW
|
9.3 | Ki | 2 | — | |
IFPPYSWJNWHOLQ
|
9.3 | Ki | 52 | Yes | |
KNARVZUUCLIBGV
|
9.3 | Ki | 33 | — | |
MCXANZUXLRCMDM
|
9.3 | IC50 | 2 | Yes | |
OTKXMYZOSPIKMY
|
9.3 | IC50 | 3 | — | |
UBPYILGKFZZVDX
|
9.3 | Kd | 130 | Yes | |
VOVZXURTCKPRDQ
|
9.3 | IC50 | 2 | — | |
CZCGARLOFSDTBA
|
9.3 | Ki | 2 | — | |
AXCUTSXYMWKWEA
|
9.3 | IC50 | 2 | — | |
KOIRZEHURFRWOY
|
9.3 | IC50 | 2 | — | |
WKTHEPAGRCQCOF
|
9.3 | IC50 | 2 | — | |
WTEAUFXGRKOZNT
|
9.3 | IC50 | 2 | — | |
XJPZWFIHWISMOH
|
9.3 | IC50 | 2 | — | |
LFLRMYZNGFXKMP
|
9.3 | IC50 | 2 | — | |
IALDYVNFZAPNJV
|
9.2 | IC50 | 11 | — | |
LQBDBQSMCXTVKB
|
9.2 | IC50 | 2 | — | |
MBGWSLGJUQDACI
|
9.2 | IC50 | 2 | — | |
QTYVZNNBMDNHJL
|
9.2 | IC50 | 3 | — | |
CAWFLWKFZFPVQV
|
9.2 | IC50 | 3 | — | |
MHCPAORAYMTGCZ
|
9.2 | Ki | 37 | — | |
QWKZREQFPCVBBG
|
9.2 | IC50 | 2 | — | |
MQXNKLLRIGGEOE
|
9.2 | Kd | 3 | — | |
XTFQLAOUVSZDDX
|
9.2 | IC50 | 3 | — | |
JGXRYYVIMAYABB
|
9.2 | IC50 | 2 | — | |
DFMJWYNOKUEPJT
|
9.2 | IC50 | 2 | — | |
MKHTUOFMIYFSEP
|
9.2 | Kd | 3 | — | |
SWVWXQFAJXFRCG
|
9.2 | IC50 | 3 | — | |
WHTDVCOWKCEOHS
|
9.2 | IC50 | 2 | — | |
ZVLDJWAUCMOGIZ
|
9.1 | IC50 | 2 | — | |
QXWCRBMAGJJKTO
|
9.1 | IC50 | 4 | Yes | |
ZLMYOQZUWFEOHX
|
9.1 | IC50 | 2 | — | |
NYUZAHPHSBKPPK
|
9.1 | IC50 | 3 | — | |
WCWDBZHYAHZGNZ
|
9.1 | IC50 | 3 | — | |
XHORJSJFHVABEA
|
9.1 | Ki | 5 | — | |
XHORJSJFHVABEA
|
9.1 | Ki | 49 | — | |
PHXJVRSECIGDHY
|
9.1 | IC50 | 59 | — | |
ZQOBVMHBVWNVBG
|
9.1 | IC50 | 2 | — | |
AYQXKPMEHPZRKR
|
9.0 | IC50 | 6 | — | |
JTWMOWRMSZZHDR
|
9.0 | IC50 | 13 | — | |
VGHMNDGFXSTBOE
|
9.0 | Kd | 3 | — | |
RZOMPFGUSZPJBC
|
9.0 | IC50 | 3 | — | |
ZBNZXTGUTAYRHI
|
9.0 | IC50 | 102 | Yes | |
NUTAFQYFQXUSOF
|
9.0 | IC50 | 2 | — | |
AJVISBGKRJRTQV
|
9.0 | Ki | 2 | — | |
BNRXMSGHPVYSDK
|
9.0 | IC50 | 24 | — | |
CRLZGLXSANQWFT
|
9.0 | IC50 | 6 | — | |
KZYSNMDDKMTSHZ
|
9.0 | IC50 | 3 | — | |
QZGWWTNGPOKJGC
|
9.0 | IC50 | 2 | — | |
SLCFEJAMCRLYRG
|
9.0 | Kd | 8 | Yes |