Target Details
| UniProt AC | P00519 |
|---|---|
| Gene Symbol | ABL1 |
| Protein Name | Tyrosine-protein kinase ABL1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08919 (F_actin_bind) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,419
- Clinical molecules 468
- Avg pChEMBL 7.25
KEGG Pathways (12)
Associated Diseases (3)
Active Molecules (1,419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YXTDYCAIPCZQMK
|
7.1 | IC50 | 3 | — | |
ZAXFYYCHCGZIPG
|
7.1 | IC50 | 2 | — | |
AZCFXTPLBWULJY
|
7.1 | IC50 | 2 | — | |
DZJWVPHWQSPJDD
|
7.1 | IC50 | 2 | — | |
FZXLZZAXHCHSEG
|
7.1 | IC50 | 2 | — | |
KAUYVUREAPHUSF
|
7.1 | IC50 | 5 | Yes | |
KEQJVXCNVVFRCN
|
7.1 | IC50 | 2 | — | |
KNGAOBKKLCKYNZ
|
7.1 | IC50 | 5 | — | |
SDYGMEWQBSWSIW
|
7.1 | IC50 | 6 | — | |
UHTHHESEBZOYNR
|
7.1 | Kd | 66 | Yes | |
LCYSSHSIKSARGO
|
7.1 | IC50 | 19 | — | |
VVLOLXBDTFEURK
|
7.1 | IC50 | 10 | Yes | |
XYFPWWZEPKGCCK
|
7.1 | IC50 | 34 | — | |
YZLKFFPFWYDBEB
|
7.1 | IC50 | 3 | — | |
CXUFYCPSBOYQMV
|
7.0 | IC50 | 5 | — | |
JONUUBFCZUAOFY
|
7.0 | IC50 | 10 | — | |
KUUKOPMICNKRGE
|
7.0 | IC50 | 12 | Yes | |
NBRVSSMSYRPVCE
|
7.0 | Ki | 2 | Yes | |
OVPLBDSXFCRGJY
|
7.0 | IC50 | 5 | Yes | |
SRTONYAWGLMSSN
|
7.0 | IC50 | 4 | Yes | |
UEVPEEHDLTWCMS
|
7.0 | Ki | 3 | Yes | |
XNWHPCMDUYIUSL
|
7.0 | Ki | 2 | Yes | |
HKSZLNNOFSGOKW
|
7.0 | Kd | 408 | — | |
NQRWHNMIXKRPES
|
7.0 | IC50 | 2 | — | |
RGUQJUZAJQPBOS
|
7.0 | IC50 | 3 | — | |
UWHYTXRXDYNHKS
|
7.0 | IC50 | 3 | — | |
WHPAIRPZLHBOIC
|
7.0 | Ki | 3 | Yes | |
VZHQCVYEVMECQT
|
7.0 | IC50 | 2 | — | |
BYKVUESQXQHBEP
|
7.0 | IC50 | 7 | — | |
FRSWPGKMMGVEGT
|
7.0 | IC50 | 2 | — | |
QGLVSYZUEILELT
|
7.0 | IC50 | 3 | — | |
QMCPPBRAJKQPLH
|
7.0 | IC50 | 3 | — | |
RQMAVXSBMSSQDJ
|
7.0 | IC50 | 3 | — | |
HRCGOBVLZLYNFI
|
7.0 | IC50 | 2 | — | |
KTEIFNKAUNYNJU
|
7.0 | Kd | 114 | — | |
PKDOQGUKLRAMEF
|
7.0 | IC50 | 3 | — | |
WJSCDYSIDGEWEB
|
7.0 | IC50 | 5 | Yes | |
YYIDVDRESUYFKM
|
7.0 | IC50 | 3 | — | |
CNTCGRJDUJEUDG
|
7.0 | Ki | 37 | — | |
DLWMVUDMPMKGEE
|
7.0 | Ki | 24 | — | |
DZHIOWDUNSAQDE
|
7.0 | IC50 | 2 | — | |
HKSZLNNOFSGOKW
|
7.0 | Ki | 118 | — | |
HUNGUWOZPQBXGX
|
7.0 | IC50 | 4 | — | |
JHMBUEWQJDGKGS
|
7.0 | IC50 | 7 | Yes | |
LVOBTCONHRNJJA
|
7.0 | IC50 | 4 | Yes | |
MVJMMLFMPWITEJ
|
7.0 | Ki | 110 | — | |
OBLBAQUXHOPUQG
|
7.0 | IC50 | 3 | — | |
OIMJFVHFGBCRHO
|
7.0 | IC50 | 2 | — | |
PGYXMFATLWTNBT
|
7.0 | Ki | 3 | Yes | |
PIQCTGMSNWUMAF
|
7.0 | Kd | 137 | Yes |