Target Details
| UniProt AC | P00519 |
|---|---|
| Gene Symbol | ABL1 |
| Protein Name | Tyrosine-protein kinase ABL1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08919 (F_actin_bind) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,419
- Clinical molecules 468
- Avg pChEMBL 7.25
KEGG Pathways (12)
Associated Diseases (3)
Active Molecules (1,419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IORXBTIJLGQAEJ
|
7.2 | IC50 | 2 | — | |
FGMSUCIOAMNCKF
|
7.2 | IC50 | 3 | Yes | |
OSZVHJYNXBUVAH
|
7.2 | IC50 | 12 | — | |
RHFWTFDTRBFIHU
|
7.2 | IC50 | 13 | Yes | |
XNODQMMIMXSTMX
|
7.2 | IC50 | 12 | Yes | |
CQWRMHYRBJWJNS
|
7.2 | IC50 | 5 | — | |
FAWGCSGOLCHXBH
|
7.2 | IC50 | 11 | Yes | |
GXMFPDCIAWSZFR
|
7.2 | IC50 | 5 | — | |
MQBBZKCWIDFMIQ
|
7.2 | Ki | 3 | Yes | |
MWYBBCLGEHZSCP
|
7.2 | IC50 | 11 | Yes | |
MZVPLRQASMAJIS
|
7.2 | IC50 | 3 | Yes | |
PANUCCHSDROJBK
|
7.2 | IC50 | 3 | — | |
QEKCMFKWDZHOOD
|
7.2 | IC50 | 6 | Yes | |
USMCKQQKWYXXCV
|
7.2 | IC50 | 2 | — | |
ZFTWKPRQHPMJAA
|
7.2 | IC50 | 2 | — | |
GXAIYZPLZBVGNJ
|
7.2 | IC50 | 3 | — | |
QHNQSGOQPWOVDK
|
7.2 | IC50 | 2 | — | |
BFSMWDPRHAHFSS
|
7.1 | IC50 | 2 | — | |
FHNLPTRXVQOXQO
|
7.1 | IC50 | 11 | Yes | |
IQPVVCXHSILADO
|
7.1 | IC50 | 3 | Yes | |
JHOCOYLYGFKRLD
|
7.1 | Ki | 3 | Yes | |
QQWUGDVOUVUTOY
|
7.1 | Kd | 231 | Yes | |
VOYZWDQJVPQGCO
|
7.1 | IC50 | 9 | — | |
WQIKRJDLIIEKAG
|
7.1 | IC50 | 2 | — | |
HRKJFKJZUNJKNU
|
7.1 | IC50 | 10 | — | |
IDMLCHSTWFWJHX
|
7.1 | IC50 | 2 | — | |
CBWWAMHIIZVQTP
|
7.1 | IC50 | 6 | — | |
RXNGGTYNZUEFOM
|
7.1 | IC50 | 8 | Yes | |
SMPGEBOIKULBCT
|
7.1 | IC50 | 15 | — | |
XXJWYDDUDKYVKI
|
7.1 | Kd | 52 | — | |
AYYRUOOCJNTWHJ
|
7.1 | IC50 | 5 | — | |
DBXOMQJZSQLQED
|
7.1 | Ki | 12 | — | |
DDRLQMSTWJRCMI
|
7.1 | IC50 | 2 | — | |
FQYLJBVSYHZWLT
|
7.1 | Ki | 35 | Yes | |
HXHAJRMTJXHJJZ
|
7.1 | Ki | 52 | Yes | |
IBPVXAOOVUAOKJ
|
7.1 | IC50 | 5 | — | |
KFUPFXKVTHKTDP
|
7.1 | IC50 | 2 | — | |
KTEIFNKAUNYNJU
|
7.1 | Ki | 48 | — | |
KVXUSGCDEMAYHI
|
7.1 | Ki | 4 | — | |
MQRDVGBWWVWMEN
|
7.1 | Ki | 47 | — | |
NSYXCWYWACQNOH
|
7.1 | Ki | 10 | — | |
PSKGMHXAYOCLLX
|
7.1 | IC50 | 2 | — | |
QNYNFUREPOMYSY
|
7.1 | Ki | 3 | Yes | |
RGNHKJWHFIPHIM
|
7.1 | Ki | 66 | — | |
VNGYQBMDQMDALH
|
7.1 | Ki | 25 | — | |
GKLDJIUKRHJMHG
|
7.1 | IC50 | 2 | — | |
YJNVZAXZUDOAAI
|
7.1 | IC50 | 10 | Yes | |
AACFRJDPYQPXPD
|
7.1 | Ki | 3 | Yes | |
CHLFFSKXUJQLQO
|
7.1 | IC50 | 7 | — | |
OGFUMLMDBRBYKQ
|
7.1 | IC50 | 3 | — |