Target Details
| UniProt AC | P00519 |
|---|---|
| Gene Symbol | ABL1 |
| Protein Name | Tyrosine-protein kinase ABL1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08919 (F_actin_bind) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,419
- Clinical molecules 468
- Avg pChEMBL 7.25
KEGG Pathways (12)
Associated Diseases (3)
Active Molecules (1,419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NYEBJLYZEHKODB
|
7.4 | Ki | 5 | Yes | |
PPMFZQWMHKWFPZ
|
7.4 | IC50 | 2 | — | |
ZMQAYSHYLVAIDP
|
7.4 | IC50 | 2 | — | |
JIBBGYSUSKAPDY
|
7.4 | IC50 | 19 | — | |
RWKFWKPIQLFUQP
|
7.4 | IC50 | 6 | — | |
YQXVNNKJNHKVLW
|
7.4 | Kd | 3 | — | |
NPQDLAMGUSTRMY
|
7.4 | IC50 | 3 | — | |
XEXBRZPNVDDJRA
|
7.4 | IC50 | 2 | — | |
YSFGCARYACLFDS
|
7.4 | Ki | 7 | Yes | |
YTOXAXYCYYWBRD
|
7.4 | IC50 | 2 | — | |
LVUGPVDXTSJQQD
|
7.3 | IC50 | 13 | Yes | |
ONYASORTFKFDEA
|
7.3 | IC50 | 2 | — | |
AGENIADQYCDWLP
|
7.3 | IC50 | 3 | — | |
DQHVUKLVCBJBLM
|
7.3 | IC50 | 8 | — | |
JXXVUIBYJYNDBA
|
7.3 | IC50 | 3 | — | |
QOHRZEWGDUREJV
|
7.3 | IC50 | 2 | — | |
UKHOXYCPBAGGAN
|
7.3 | Kd | 3 | — | |
VPZGFKSLFAEGRG
|
7.3 | IC50 | 2 | — | |
ADGOPPKEIZXKAZ
|
7.3 | IC50 | 3 | — | |
HFGUPJNHEPCEHX
|
7.3 | IC50 | 3 | — | |
MBNGMHXKMKQYBP
|
7.3 | Ki | 3 | Yes | |
CXQHYVUVSFXTMY
|
7.3 | Kd | 154 | — | |
LNPOXTZTOXVGTM
|
7.3 | IC50 | 3 | Yes | |
PGQWALGGBUYLQF
|
7.3 | IC50 | 12 | — | |
QRDCOOSKIFYKIQ
|
7.3 | IC50 | 8 | — | |
DHKJMXHLKKNTKJ
|
7.3 | IC50 | 5 | Yes | |
PCQMERRARZKTPW
|
7.3 | Ki | 68 | — | |
QXRJBJVCBQSLTA
|
7.3 | Ki | 29 | — | |
SDBOIBYRBWPIEL
|
7.3 | Ki | 31 | — | |
SMFAJPHTYQUDOC
|
7.3 | IC50 | 5 | Yes | |
TWCOARREJINKIL
|
7.3 | IC50 | 2 | — | |
WVFIZRNACLGJDI
|
7.3 | IC50 | 2 | — | |
XNEPVLVYFUGJLF
|
7.3 | Ki | 27 | — | |
ZLVOTRRGLSDLPF
|
7.3 | Ki | 36 | — | |
UMBFDGUGXMOMHX
|
7.3 | IC50 | 12 | — | |
UUUZEMLVABCSCR
|
7.3 | IC50 | 3 | — | |
WYQRWWCPRIGMCS
|
7.3 | IC50 | 6 | — | |
CAAAKLVRRGRQHX
|
7.3 | IC50 | 3 | — | |
MJALZBJFTIQSSR
|
7.3 | IC50 | 12 | Yes | |
NFCXPDAZPBFBRT
|
7.3 | IC50 | 3 | — | |
OFBWCZMTFNTSHE
|
7.3 | IC50 | 3 | — | |
SQQPRORGDVPLSI
|
7.3 | IC50 | 4 | — | |
TYVQJCSBHJOJCN
|
7.3 | IC50 | 2 | — | |
UARVSLPFGRKWQN
|
7.3 | IC50 | 11 | — | |
NMCRRFLWJZUPRE
|
7.3 | IC50 | 5 | Yes | |
ORTYQHFTTCRJIP
|
7.3 | IC50 | 2 | — | |
BCZRYISUUHVFEC
|
7.3 | IC50 | 2 | — | |
CFTUNRCBCCNBLL
|
7.3 | IC50 | 2 | — | |
COWHLOGPEGRMOS
|
7.3 | IC50 | 2 | — | |
JAXPOXBSVKSIEC
|
7.3 | IC50 | 2 | — |