Target Details
| UniProt AC | P00519 |
|---|---|
| Gene Symbol | ABL1 |
| Protein Name | Tyrosine-protein kinase ABL1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08919 (F_actin_bind) PF07714 (PK_Tyr_Ser-Thr) PF00017 (SH2) PF00018 (SH3_1) |
Summary
- Multi-target molecules 1,419
- Clinical molecules 468
- Avg pChEMBL 7.25
KEGG Pathways (12)
Associated Diseases (3)
Active Molecules (1,419)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BTIKYUUNPGWLNG
|
7.5 | IC50 | 12 | Yes | |
OKHCJZLKVVFPLZ
|
7.5 | IC50 | 2 | — | |
CQBBMNXXVMOFCA
|
7.5 | Ki | 39 | — | |
NWKLIKWHLFEAFY
|
7.5 | IC50 | 2 | — | |
PTVPBWWDGZSEAF
|
7.5 | Ki | 63 | — | |
UIQVTQZGYNQWLN
|
7.5 | IC50 | 2 | — | |
VEORWCZDRQSGJH
|
7.5 | IC50 | 10 | Yes | |
DFYOVMKHYAWORB
|
7.5 | IC50 | 3 | Yes | |
JKZZCHSVFXZBAI
|
7.5 | IC50 | 6 | — | |
SSDFTYWIYVWCIE
|
7.5 | IC50 | 17 | — | |
DUJMHEBMAPADNS
|
7.5 | IC50 | 4 | — | |
FJLUYTVEVSZLJP
|
7.5 | IC50 | 5 | — | |
RIXBMLAVFFOVIP
|
7.5 | IC50 | 2 | — | |
UESYKRUJFLCOLW
|
7.5 | IC50 | 5 | — | |
AKRIJSSBKYPXID
|
7.5 | IC50 | 3 | — | |
WFQCEVIDLOLEDG
|
7.5 | IC50 | 5 | — | |
FYTNSFVHUFSPDY
|
7.5 | IC50 | 3 | — | |
IWODHENDABKBRB
|
7.5 | IC50 | 6 | — | |
JJFYUQKAJYRNHL
|
7.5 | IC50 | 2 | — | |
NMMIVVLEPHGUEV
|
7.5 | IC50 | 2 | — | |
OATHVDKMFZZHHN
|
7.5 | IC50 | 9 | — | |
MXJMJNRCJKHFPP
|
7.4 | IC50 | 10 | — | |
QDXRELOFIZDHGS
|
7.4 | IC50 | 2 | — | |
RITAVMQDGBJQJZ
|
7.4 | Kd | 43 | — | |
INHKTKGJEIKALZ
|
7.4 | IC50 | 2 | — | |
RHWUJWQTWHXYPV
|
7.4 | IC50 | 3 | — | |
XQKRNUCXAFMEFO
|
7.4 | IC50 | 3 | — | |
BYODDABQBNBRRN
|
7.4 | IC50 | 2 | — | |
JWDIICDIOIJDNV
|
7.4 | IC50 | 2 | — | |
KILAESXRGZQREB
|
7.4 | IC50 | 3 | Yes | |
XPWYQHDVNYIXSF
|
7.4 | IC50 | 2 | — | |
YCFQNCQMGGRGHM
|
7.4 | IC50 | 4 | Yes | |
YTHUQGIGAIZNIM
|
7.4 | IC50 | 3 | — | |
CSGDMICHMNNVRM
|
7.4 | IC50 | 2 | — | |
CAHQAXRCSXNZRF
|
7.4 | IC50 | 5 | Yes | |
DAZCBQNFGSWSQG
|
7.4 | IC50 | 8 | Yes | |
HKZKELVPGXJIMW
|
7.4 | Ki | 41 | — | |
HXPKYBPDEWUZKU
|
7.4 | IC50 | 3 | — | |
IDZXNZQRVWDXGU
|
7.4 | Ki | 3 | Yes | |
KSCBSHLEWGZVON
|
7.4 | IC50 | 4 | — | |
LVECPYVAIBNSRV
|
7.4 | Ki | 33 | — | |
SEJGTFPOEJWEGG
|
7.4 | Kd | 149 | — | |
SHTNULLAAVPXRC
|
7.4 | IC50 | 4 | — | |
VISDQUKQUGPQNV
|
7.4 | IC50 | 5 | Yes | |
ZCXFAEZLYWAZMY
|
7.4 | Ki | 3 | Yes | |
QAOMWMNQOYMGAR
|
7.4 | IC50 | 2 | — | |
QCUODDVWGHBDKJ
|
7.4 | IC50 | 3 | — | |
QXLGSVJYRNECIT
|
7.4 | IC50 | 3 | — | |
VSCYVMFGKQHZQG
|
7.4 | IC50 | 3 | — | |
XLMBXWNZLPFUQW
|
7.4 | IC50 | 2 | — |