Target Details
| UniProt AC | P00469 |
|---|---|
| Gene Symbol | thyA |
| Protein Name | Thymidylate synthase |
| Organism | Lacticaseibacillus casei |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00303 (Thymidylat_synt) |
Summary
- Multi-target molecules 26
- Clinical molecules 10
- Avg pChEMBL 7.64
Active Molecules (26)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HUEGPYLGWYYQEQ
|
10.0 | Ki | 2 | — | |
VPWDSJXYLFJZOZ
|
8.8 | Ki | 2 | — | |
FBOZXECLQNJBKD
|
8.6 | IC50 | 16 | — | |
WENVMKCBNUSGID
|
8.6 | IC50 | 2 | — | |
NFARHPAOOHOWAL
|
8.4 | IC50 | 2 | — | |
LTKHPMDRMUCUEB
|
8.1 | IC50 | 2 | — | |
YVHACGQTVJQBQW
|
7.9 | IC50 | 3 | — | |
YVHACGQTVJQBQW
|
7.9 | IC50 | 3 | Yes | |
CUZJGZKZBQUBIR
|
7.8 | IC50 | 3 | — | |
CUZJGZKZBQUBIR
|
7.8 | IC50 | 3 | Yes | |
KAYSCGYEDLPRGH
|
7.8 | IC50 | 3 | — | |
KAYSCGYEDLPRGH
|
7.8 | IC50 | 3 | Yes | |
UUVHCWYURYQGNG
|
7.8 | IC50 | 3 | — | |
UUVHCWYURYQGNG
|
7.8 | IC50 | 3 | Yes | |
DSIACOJIIGFHHZ
|
7.7 | IC50 | 2 | — | |
OMHZMMMKMRPSKH
|
7.7 | IC50 | 3 | Yes | |
SNCKXYAIQODZOE
|
7.7 | IC50 | 3 | — | |
SNCKXYAIQODZOE
|
7.7 | IC50 | 3 | Yes | |
UWMZMPSPAFBAOA
|
7.7 | IC50 | 2 | — | |
LTKHPMDRMUCUEB
|
7.3 | IC50 | 4 | Yes | |
AOGOUTMDEVCZHA
|
6.8 | IC50 | 3 | Yes | |
XYVUDAYNSCLZJK
|
6.5 | IC50 | 2 | — | |
WBXPDJSOTKVWSJ
|
6.3 | Ki | 10 | Yes | |
RJTQNRRVLFIIEV
|
6.0 | Ki | 2 | Yes | |
BJJFDFPYWNZIKB
|
6.0 | Ki | 2 | — | |
VVUKQBRYAJFWQT
|
6.0 | IC50 | 2 | — |