Target Details
UniProt ACP00382
Gene SymboldhfrI
Protein NameDihydrofolate reductase type 1
OrganismEscherichia coli
Entry Name
Organism Category Pathogen
Pfam Domains PF00186 (DHFR_1)
Summary
  • Multi-target molecules 36
  • Clinical molecules 0
  • Avg pChEMBL 7.01
Top Co-occurrence Targets
Active Molecules (36)
InChIKey pChEMBL Type Targets Clinical
HKVFBDOFZVZRHQ 8.7 IC50 3
ROFHCHDLNGIYAX 8.6 IC50 2
VFMMMIYNLXXETQ 8.2 IC50 2
IUTSNRRXQPUZNH 8.1 IC50 2
FGMLPHRAADCMBM 8.0 Ki 2
AAMMQVFLCXMBIO 8.0 Ki 2
IZJHXNMVMRCLAW 7.9 IC50 2
MMPFYSRMKOTYDR 7.8 IC50 2
WKFJKDHKBGEBJS 7.8 Ki 3
NMARPFMJVCXSAV 7.7 Ki 4
PXEPXKJNUDMGFE 7.7 IC50 2
VOABTGRNIMDWHY 7.5 IC50 2
KUPCVEUDIMEMHK 7.4 IC50 2
QBQZTCRZECEEGK 7.3 Ki 3
AEQAPJCADMGBFW 7.2 IC50 2
BVTLYXPJXLFKHC 7.1 IC50 2
YBIRDHJXPIORJB 7.1 Ki 3
FKTRXRCVRZPVFR 6.9 Ki 2
DMGSYGBIKYHPEJ 6.9 IC50 2
NTVMHTFWSNGDLC 6.9 Ki 4
VZDZIQCTRIYVLF 6.8 IC50 2
LMWNROFCHOPQFZ 6.6 Ki 3
YZGBAURBIITWIY 6.6 Ki 3
IEDVJHCEMCRBQM 6.3 IC50 7
RWXWLTHUGRWMRC 6.3 Ki 3
AIZLSGCCJQCUJL 6.2 Ki 3
QPXDTEXOMMULLS 6.2 Ki 3
XHJNBBKNRVVKOH 6.2 Ki 3
SJLUGNSWLCFURF 6.2 Ki 2
KLTBXEYFWQXDEU 6.2 Ki 2
IHLMFJNDHCQZGA 6.1 Ki 2
UHSFYDTWKATRPP 6.0 Ki 3
VRXFDHXUFJMNEH 6.0 Ki 3
ZJKYATYSNJZLSA 6.0 Ki 3
HDNCDAIQTLSPPL 6.0 Ki 3
JEJKECLVSUQMHZ 6.0 Ki 3
2D structure