Target Details
| UniProt AC | P00381 |
|---|---|
| Gene Symbol | folA |
| Protein Name | Dihydrofolate reductase |
| Organism | Lacticaseibacillus casei |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00186 (DHFR_1) |
Summary
- Multi-target molecules 65
- Clinical molecules 2
- Avg pChEMBL 7.56
Active Molecules (65)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QBQZTCRZECEEGK
|
6.5 | Ki | 3 | — | |
LMWNROFCHOPQFZ
|
6.5 | Ki | 3 | — | |
IHLMFJNDHCQZGA
|
6.5 | Ki | 2 | — | |
AAMMQVFLCXMBIO
|
6.4 | Ki | 2 | — | |
UHSFYDTWKATRPP
|
6.4 | Ki | 3 | — | |
FXGBKUVTNNFJHR
|
6.4 | IC50 | 2 | — | |
NTVMHTFWSNGDLC
|
6.3 | Ki | 4 | — | |
YBIRDHJXPIORJB
|
6.3 | Ki | 3 | — | |
VEBQFPSIZLJALQ
|
6.3 | Ki | 2 | — | |
ACXZKUHGYNILFP
|
6.2 | IC50 | 3 | — | |
ACXZKUHGYNILFP
|
6.2 | IC50 | 3 | — | |
RYPITQKKMGHSMZ
|
6.1 | Ki | 2 | — | |
JHSUWQJDEDXPGP
|
6.0 | IC50 | 2 | — | |
AIZLSGCCJQCUJL
|
6.0 | Ki | 3 | — | |
DGQWEZFLVCMZJD
|
6.0 | Ki | 3 | — |