Target Details
| UniProt AC | O96020 |
|---|---|
| Gene Symbol | CCNE2 |
| Protein Name | G1/S-specific cyclin-E2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) |
Summary
- Multi-target molecules 504
- Clinical molecules 252
- Avg pChEMBL 7.06
KEGG Pathways (17)
- Cell cycle
- Cellular senescence
- Cushing syndrome
- Epstein-Barr virus infection
- Gastric cancer
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Measles
- MicroRNAs in cancer
- Oocyte meiosis
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (504)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PMXCMJLOPOFPBT
|
7.5 | IC50 | 17 | Yes | |
UVLBAPBHAHFJSY
|
7.5 | IC50 | 8 | Yes | |
DGPWUICUWDZQNV
|
7.4 | IC50 | 7 | Yes | |
DXVKJMDIJODFKP
|
7.4 | IC50 | 5 | Yes | |
HEFHQIBQGOCQAF
|
7.4 | IC50 | 11 | Yes | |
SJTMBARMWBHQAM
|
7.4 | IC50 | 3 | — | |
XACARXKEKLHSQO
|
7.4 | IC50 | 5 | Yes | |
XNKBKFNLOYVTSF
|
7.4 | IC50 | 11 | — | |
SVZUZSDHGKVQNU
|
7.4 | IC50 | 11 | Yes | |
UMJDAZSXABEMLH
|
7.4 | IC50 | 4 | — | |
BBNBFSYCPUPPCC
|
7.4 | IC50 | 5 | — | |
MHSDRURPTIXMJZ
|
7.4 | IC50 | 5 | — | |
POARIJJCCJDSKV
|
7.4 | IC50 | 5 | Yes | |
QNKYOKCOZLJDJO
|
7.4 | IC50 | 3 | — | |
SUEYMQKVBANZMC
|
7.4 | IC50 | 8 | Yes | |
YYJIVPXZKPNMQZ
|
7.4 | IC50 | 5 | Yes | |
STWGJFWWXVBMEE
|
7.4 | IC50 | 5 | Yes | |
KZIAOAADZPTJQN
|
7.4 | Ki | 4 | — | |
BYPSHOOZDMABOO
|
7.4 | IC50 | 5 | Yes | |
CNXYYBLJBYUISF
|
7.4 | IC50 | 3 | — | |
OUNCSFZWBHZJNV
|
7.3 | IC50 | 3 | — | |
KWNRFWAMLDHJIJ
|
7.3 | IC50 | 3 | — | |
JTVILUUAQWQWBK
|
7.3 | IC50 | 8 | Yes | |
OUSFTKFNBAZUKL
|
7.3 | IC50 | 58 | Yes | |
RABZCZVASTTWML
|
7.3 | IC50 | 5 | Yes | |
HOEMOEJHHVVLJW
|
7.3 | IC50 | 8 | Yes | |
JGNMMLNIOWYNHJ
|
7.3 | IC50 | 8 | — | |
KVNDPOMKLVNLRR
|
7.3 | IC50 | 3 | — | |
NGLJEWVPKWMIAJ
|
7.3 | IC50 | 5 | — | |
SCAGLYMBBLMFND
|
7.3 | IC50 | 8 | Yes | |
SVGBMXDLMHCYLQ
|
7.3 | IC50 | 3 | — | |
VFUZGZRCARGQHE
|
7.3 | IC50 | 3 | — | |
VVXLHYKOWIXRSV
|
7.3 | IC50 | 5 | — | |
ZIXQXEIXOHWQCK
|
7.3 | IC50 | 3 | — | |
CNNQBAXDFGTALM
|
7.3 | IC50 | 5 | — | |
GTAZDNZBVNYMQW
|
7.3 | IC50 | 3 | — | |
UAOIPNOTWOYAMU
|
7.3 | IC50 | 11 | Yes | |
VSFMTQXQSZZVEU
|
7.3 | IC50 | 5 | Yes | |
XAKCLNJQGRBKPQ
|
7.3 | IC50 | 5 | — | |
AMZVBIHYDIQGRK
|
7.2 | Ki | 4 | — | |
DOHWEZMWGPLSGI
|
7.2 | IC50 | 5 | Yes | |
ZEHXSPZMRLUPSR
|
7.2 | IC50 | 7 | Yes | |
FIZSPBCJAWUURL
|
7.2 | IC50 | 3 | — | |
NHCOZCJPPTVVOW
|
7.2 | IC50 | 7 | Yes | |
YUOUZNKMAFVMNY
|
7.2 | IC50 | 3 | — | |
DYGQMQPINIGYEV
|
7.2 | IC50 | 5 | Yes | |
JWYXJDKUBNYUOI
|
7.2 | IC50 | 3 | — | |
RHOFDJKXENXNLN
|
7.2 | IC50 | 7 | Yes | |
UIAYOLLUEZBQEH
|
7.2 | IC50 | 6 | — | |
VQWRERKTQFNERF
|
7.2 | IC50 | 8 | — |