Target Details
| UniProt AC | O96020 |
|---|---|
| Gene Symbol | CCNE2 |
| Protein Name | G1/S-specific cyclin-E2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) |
Summary
- Multi-target molecules 504
- Clinical molecules 252
- Avg pChEMBL 7.06
KEGG Pathways (17)
- Cell cycle
- Cellular senescence
- Cushing syndrome
- Epstein-Barr virus infection
- Gastric cancer
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Measles
- MicroRNAs in cancer
- Oocyte meiosis
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (504)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PIDYSPIUVLYIJV
|
7.8 | IC50 | 5 | Yes | |
XSAPHSITEDFKJO
|
7.8 | IC50 | 3 | — | |
CVBCPFYFIGQTLV
|
7.7 | IC50 | 3 | — | |
HZELJXXPCYGOOL
|
7.7 | IC50 | 9 | Yes | |
IAEDTIBMQBGVIX
|
7.7 | IC50 | 5 | Yes | |
MKQRMAQXDANGMN
|
7.7 | IC50 | 8 | Yes | |
NQZLCGLQVAVSGY
|
7.7 | IC50 | 4 | — | |
NRCIGJZLDFFIDD
|
7.7 | IC50 | 8 | Yes | |
OSCCTZDFBLPFFT
|
7.7 | IC50 | 5 | Yes | |
TYIGVUBZPQNYTD
|
7.7 | IC50 | 4 | Yes | |
TZSZKILLRMGQIE
|
7.7 | IC50 | 5 | Yes | |
VDOFFDSHVJGCSN
|
7.7 | IC50 | 5 | Yes | |
WMKCACSJDBTUJB
|
7.7 | IC50 | 3 | — | |
YBLCOFFOEGGLGV
|
7.7 | IC50 | 3 | — | |
ZWVNPBSQSAHHNR
|
7.7 | IC50 | 11 | Yes | |
DJEJXDSNSASKPZ
|
7.7 | IC50 | 3 | — | |
FZLZLIAOYSKHJC
|
7.7 | Ki | 11 | — | |
IISWHFMSGFZNGY
|
7.7 | IC50 | 3 | — | |
VEZVYTFKYSTCLC
|
7.7 | IC50 | 3 | — | |
YADWBXSXYFLZKW
|
7.7 | IC50 | 5 | Yes | |
LKPJCXVMXCWQKG
|
7.7 | IC50 | 5 | Yes | |
PRXRQGZKWMOFLL
|
7.7 | IC50 | 11 | Yes | |
QXHLCISVAQTGNJ
|
7.7 | IC50 | 5 | Yes | |
SXBXZPMHHKFUPC
|
7.6 | IC50 | 5 | Yes | |
ZUCAWWSJZRVUAX
|
7.6 | Ki | 11 | — | |
CGJRRFJDMMUHJW
|
7.6 | IC50 | 5 | Yes | |
FGLRSCIZYHXTBC
|
7.6 | IC50 | 9 | Yes | |
NJCYRPYWLUDPJX
|
7.6 | IC50 | 3 | — | |
QUDNAUWPTMNNHI
|
7.6 | IC50 | 8 | Yes | |
CMNKHKYPFIVLLC
|
7.6 | IC50 | 5 | Yes | |
DJEJXDSNSASKPZ
|
7.6 | IC50 | 3 | — | |
UDGMVUGWIIYQOU
|
7.6 | IC50 | 5 | Yes | |
UFQIHIBAMFVYOW
|
7.6 | IC50 | 3 | — | |
UQBQAVMSJUVQLF
|
7.6 | IC50 | 5 | Yes | |
KHLSGMMGWBAAOY
|
7.6 | IC50 | 11 | Yes | |
KMHNZVWSMBCPMT
|
7.6 | IC50 | 8 | — | |
CFHPOEFRHPSTGX
|
7.5 | IC50 | 5 | Yes | |
PDHGOPVHZSWSKJ
|
7.5 | IC50 | 4 | Yes | |
AJIAGOODOUPWJG
|
7.5 | IC50 | 5 | Yes | |
CKUFTNKWKUUZBS
|
7.5 | IC50 | 5 | Yes | |
KBQFJASPKOEHLK
|
7.5 | IC50 | 5 | Yes | |
KFQUFRTZLXDXFK
|
7.5 | IC50 | 5 | Yes | |
LXYGBCHGOVEYQM
|
7.5 | IC50 | 8 | Yes | |
RAUGKKGXYWWHFL
|
7.5 | IC50 | 8 | Yes | |
VPYBDMKXOBHEPY
|
7.5 | IC50 | 5 | Yes | |
WRKQTFCCJAMNGR
|
7.5 | IC50 | 5 | — | |
XKWGQYSHLNEUOC
|
7.5 | IC50 | 5 | Yes | |
QARVJSXJBXBDLJ
|
7.5 | IC50 | 5 | Yes | |
ITGHQSNMEJUHKF
|
7.5 | IC50 | 5 | Yes | |
PVXGUOAMKJRLQU
|
7.5 | IC50 | 5 | Yes |