Target Details
| UniProt AC | O96020 |
|---|---|
| Gene Symbol | CCNE2 |
| Protein Name | G1/S-specific cyclin-E2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02984 (Cyclin_C) PF00134 (Cyclin_N) |
Summary
- Multi-target molecules 504
- Clinical molecules 252
- Avg pChEMBL 7.06
KEGG Pathways (17)
- Cell cycle
- Cellular senescence
- Cushing syndrome
- Epstein-Barr virus infection
- Gastric cancer
- Hepatitis B
- Human T-cell leukemia virus 1 infection
- Human papillomavirus infection
- Measles
- MicroRNAs in cancer
- Oocyte meiosis
- PI3K-Akt signaling pathway
- Pathways in cancer
- Prostate cancer
- Small cell lung cancer
- Viral carcinogenesis
- p53 signaling pathway
Associated Diseases (1)
Active Molecules (504)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IKQWJXXGBHAZAL
|
8.1 | IC50 | 5 | Yes | |
IQFWZWLHQMBGKM
|
8.1 | IC50 | 5 | Yes | |
KAFOMMCZXZCPNQ
|
8.1 | IC50 | 5 | Yes | |
NSGQRIPFMLCLFH
|
8.1 | IC50 | 8 | Yes | |
QBQOHKFVYIDSIJ
|
8.1 | IC50 | 6 | Yes | |
SCFMWQIQBVZOQR
|
8.1 | IC50 | 14 | Yes | |
YUDOGLCZMQACFU
|
8.1 | IC50 | 3 | — | |
ZKDXRFMOHZVXSG
|
8.1 | IC50 | 13 | Yes | |
AOPVKMUMEMDUCK
|
8.0 | IC50 | 8 | Yes | |
AQJSWLPZCPUBBH
|
8.0 | IC50 | 5 | Yes | |
BSDJIQDLIJZWHF
|
8.0 | IC50 | 8 | Yes | |
CQRTXGVZEGGYSB
|
8.0 | IC50 | 5 | Yes | |
FJOZRBWUECWIBB
|
8.0 | IC50 | 9 | Yes | |
FZTUTRSHORYMBR
|
8.0 | IC50 | 9 | Yes | |
HAJAIWADCDXZLK
|
8.0 | IC50 | 5 | Yes | |
HZYXPGRTGHXHTP
|
8.0 | IC50 | 5 | Yes | |
JNWVFIUTIMINMS
|
8.0 | IC50 | 3 | — | |
JRQGLWAUSPBBHJ
|
8.0 | IC50 | 5 | Yes | |
LTBGJBWIVOIOBU
|
8.0 | IC50 | 3 | — | |
MFBZGLIBOANTMZ
|
8.0 | IC50 | 5 | Yes | |
MYRDTGBYXRPRII
|
8.0 | IC50 | 8 | Yes | |
PYEYLKGWDVDOAS
|
8.0 | IC50 | 9 | Yes | |
QBBYPTLMIWFRMD
|
8.0 | IC50 | 3 | — | |
QMHDSFMOYAUERE
|
8.0 | IC50 | 5 | Yes | |
RKCYAQLWSYUIGW
|
8.0 | IC50 | 5 | Yes | |
RVQZIDJAMAEGLG
|
8.0 | IC50 | 8 | Yes | |
SUKFBTZUKNWXEF
|
8.0 | IC50 | 5 | Yes | |
UPSFNFYHUYDQAD
|
8.0 | IC50 | 5 | Yes | |
VABZZXKALNNIOQ
|
8.0 | IC50 | 5 | Yes | |
VJHPFFNCLILCCX
|
8.0 | IC50 | 3 | — | |
XKCYSUHMKZRHEL
|
8.0 | IC50 | 5 | Yes | |
ZNUCZCZYYCYWJD
|
8.0 | IC50 | 5 | Yes | |
QTTGJROYRLDUFU
|
8.0 | IC50 | 3 | — | |
BDMNMAWBZWPSJC
|
8.0 | IC50 | 9 | Yes | |
WOMVSEOJXACDOY
|
8.0 | IC50 | 5 | Yes | |
XLXZTAYYSLKIHA
|
8.0 | IC50 | 5 | Yes | |
VUCNOAQOECDGSB
|
7.9 | IC50 | 5 | Yes | |
ZBSWOVCMSGDLDX
|
7.9 | IC50 | 5 | Yes | |
AGIIDJZSMZSLJN
|
7.9 | IC50 | 9 | Yes | |
BTHSNXFROGTTCQ
|
7.9 | IC50 | 5 | Yes | |
PBKXLPOHQNEBHD
|
7.9 | IC50 | 5 | Yes | |
VLFKEQHRORLGIE
|
7.8 | IC50 | 5 | Yes | |
XNKRVQHYKHYXCS
|
7.8 | IC50 | 5 | Yes | |
HKSZLNNOFSGOKW
|
7.8 | IC50 | 408 | — | |
GEQMDKKVXALFFX
|
7.8 | Ki | 9 | — | |
HVAQMHFWXFSGJF
|
7.8 | IC50 | 8 | Yes | |
ARRBJEQXRLEBFJ
|
7.8 | IC50 | 3 | — | |
WKTFFSVUCQARKP
|
7.8 | IC50 | 8 | Yes | |
YTCCHXSWSPYPON
|
7.8 | IC50 | 5 | Yes | |
FJINXQDJHXTMEL
|
7.8 | Ki | 9 | — |